Patrick D Cunningham Niall W. A. Geraghty Patrick J. McArdle Paul V. Murphy and Timothy J. O'Sullivan pg 1; DOI: 10.1039/a604850a |
Synthesis of 1,2,4-trioxanes and 1,2,4-trioxepanes by
N-halogenosuccinimide-mediated cyclisations of unsaturated
hydroperoxyacetals
Yoshihiro Ushigoe Yoshihiro Kano and Masatomo Nojima pg 5; DOI: 10.1039/a605616d |
2-Halogeno-1,3-dithiane 1,3-dioxide: a diastereoselective carbonyl anion
equivalent in reactions with aldehydes
Varinder K. Aggarwal Giorgio Boccardo Julia M. Worrall Harry Adams and Rikki Alexander pg 11; DOI: 10.1039/a603416k |
Direct measurement of the anomeric effect in sulfoxides: conformational
analysis and X-ray crystal structures of 2-bromo- and
2-chloro-1,3-dithiane trans-1,3-dioxides
Varinder K. Aggarwal Julia M. Worrall Harry Adams Rikki Alexander and Brian F. Taylor pg 21; DOI: 10.1039/a605535d |
Generation and reaction of benzylammonium N-methylides with
N-cyanomethyl or N-(ethoxycarbonylalkyl) groups
Chen Zhang Yasuhiro Maeda Naohiro Shirai and Yoshiro Sato pg 25; DOI: 10.1039/a605337h |
Masataka Yokoyama Hirofumi Toyoshima Miyuki Shimizu and Hideo Togo pg 29; DOI: 10.1039/a604474c |
Preparation of new 2,4-disubstituted oxazoles from
N-acylaziridines
Frank W. Eastwood Patrick Perlmutter and Qi Yang pg 35; DOI: 10.1039/a604091h |
Studies on the role of conformation and of hydrogen-bonding on the
dihydroxylation of cyclic allylic alcohols: application to the synthesis
of conduritol D
Timothy J. Donohoe Peter R. Moore and Roy L. Beddoes pg 43; DOI: 10.1039/a604052g |
Synthetic approaches toward ecteinascidins. Part 1. Preparation of an
(E)-2-arylidene-3-benzyl-1,5-imino-3-benzazocin-4-one having a
protected phenol in the E-ring
Naoki Saito Kyoichi Tashiro Yukie Maru Kentaro Yamaguchi and Akinori Kubo pg 53; DOI: 10.1039/a603292c |
Stereoselective benzylic ![]() Rainer Clauss and Roger Hunter pg 71; DOI: 10.1039/a602932i |
Intramolecular photo[4+2]cycloaddition of an enone with a benzene ring
Keiki Kishikawa Satoshi Akimoto Shigeo Kohmoto Makoto Yamamoto and Kazutoshi Yamada pg 77; DOI: 10.1039/a601710j |
Intramolecular Vilsmeier processes: a new route to
cyclopenta[b]- and cyclohexa[b]-fused quinolines by
cyclisation of adipic and pimelic bis-amides
Otto Meth-Cohn and Simon Goon pg 85; DOI: 10.1039/a605294k |
Preparation and structure–chiroptical relationships of tartaric
acid-based layer-block chiral dendrimers
Hak-Fun Chow and Chi Ching Mak pg 91; DOI: 10.1039/a604539a |
Synthesis of sphingosine relatives. Part 19.1 Synthesis of
penaresidin A and B, azetidine alkaloids with actomyosin
ATPase-activating properties
Hirosato Takikawa Takeshi Maeda Masanori Seki Hiroyuki Koshino and Kenji Mori pg 97; DOI: 10.1039/a604276g |
Tandem Beckmann and Huisgen–White rearrangement of the
9-azabicyclo[3.3.1]nonan-3-one system. Part 2.1 The second
mode of the rearrangement leading to 6-(prop-1-enyl)piperidin-2-ylacetic
acid, a versatile intermediate for the syntheses of piperidine alkaloids
(+)-pinidine and (+)-monomorine I
Osamu Muraoka Bao-Zhong Zheng Kazuhito Okumura Emi Tabata Genzoh Tanabe and Michinori Kubo pg 113; DOI: 10.1039/a604266j |
The phototransformation of 5-tert-butyl-2![]() ![]() Ivan Basnak Denise McKinnell Neil Spencer Ayla Balkan Peter R. Ashton and Richard T. Walker pg 121; DOI: 10.1039/a604244i |
Use of linker for preparation of missing solid-state photoproducts:
head-to-head photodimerization of anthracene-9-propionic acid in its
crystalline double salt with cyclohexane-1,2-diamine
Yoshikatsu Ito and Gunnar Olovsson pg 127; DOI: 10.1039/a604176k |
Reactions involving fluoride ion. Part 41.1,2 Synthesis of
hexakis(trifluoromethyl)cyclopentadiene and derived cyclopentadienide
salts
Richard D. Chambers William K. Gray Julian F. S. Vaughan Stewart R. Korn Maurice Médebielle Andrei S. Batsanov Christian W. Lehmann and Judith A. K. Howard pg 135; DOI: 10.1039/a604087j |
Stereoselective synthesis of
(Z![]() ![]() ![]() ![]() Bartolo Gabriele Giuseppe Salerno Francesca De Pascali Mirco Costa and Gian Paolo Chiusoli pg 147; DOI: 10.1039/a603892a |
Use of highly stereospecific 1,3-dipolar cycloadditions of cyclic
nitrones with acetylenes in the preparation of novel heterocyclic ring
systems
W. Russell Bowman Roy V. Davies Alexandra M. Z. Slawin Gian S. Sohal Roger B. Titman and David J. Wilkins pg 155; DOI: 10.1039/a602598f |
Synthesis and reactions of reduced flavones
W. Groundwater E. Hibbs B. Hursthouse and Miklós Nyerges pg 163; DOI: 10.1039/a602245f |
Synthesis of alkylene linked bis-THA and alkylene linked benzyl-THA as
highly potent and selective inhibitors and molecular probes of
acetylcholinesterase
Yuan-Ping Pang Feng Hong Polly Quiram Tanya Jelacic and Stephen Brimijoin pg 171; DOI: 10.1039/a601642a |
Synthesis of chiral tricyclo[3.2.1.02,7]octanes by an
efficient 3-exo-trig radical cyclisation
reaction![]() Adusumilli Srikrishna and G. Veera Raghava Sharma pg 177; DOI: 10.1039/a601315e |
Facilitation of displacements at the 6-position of purines by the use of
1,4-diazabicyclo[2.2.2]octane as leaving group
Nicola K. Lembicz Sharon Grant William Clegg Roger J. Griffin Sarah L. Heath and Bernard T. Golding pg 185; DOI: 10.1039/a608207f |
Structures of Us-7 and Us-8: a new type of oxindole alkaloids isolated from
Uncaria attenuata Korth
Norio Aimi Toshikazu Shimizu Hiroyuki Sada Hiromitsu Takayama Shin-ichiro Sakai Sumphan Wongseripipatana and Dhavadee Ponglux pg 187; DOI: 10.1039/a607017e |
Facile construction of spirobicyclic skeletons by intramolecular aldol
reaction: simple formal syntheses of ()-spirojatamol and
()-erythrodiene
Yuji Tokunaga Maki Yagihashi Masataka Ihara and Keiichiro Fukumoto pg 189; DOI: 10.1039/a606151f |
Facile preparation of acetals and enol ethers derived from
1-arylpiperidin-4-ones
Montserrat Faja Colin B. Reese Quanlai Song and Pei-Zhuo Zhang pg 191; DOI: 10.1039/a606191e |
Synthesis based on cyclohexadienes. Part 21.1 Total synthesis of
()-hinesol and ()-10-epi-hinesol
Seenivasaga N. Janaki and G. S. R. Subba Rao pg 195; DOI: 10.1039/a606197d |
Conversion of imino-1,2,3-dithiazoles into 2-cyanobenzothiazoles,
cyanoimidoyl chlorides and diatomic sulfur
Russell F. English Oleg A. Rakitin Charles W. Rees and Olga G. Vlasova pg 201; DOI: 10.1039/a605815i |
A mild oxidative transformation of nitro compounds into ketones by
tetrapropylammonium perruthenate
Yuji Tokunaga Masataka Ihara and Keiichiro Fukumoto pg 207; DOI: 10.1039/a606332b |
Regio- and stereo-selective additions of sodium selenides to conjugate
enyne sulfones: a convenient synthesis of
4-seleno-1-sulfonylbuta-1,3-dienes
Mitsuhiro Yoshimatsu and Junko Hasegawa pg 211; DOI: 10.1039/a605547h |
Regioselective 1,4-addition of ammonia to 1-arylalka-1,3-dienes and
1-aryl-4-phenylbuta-1,3-dienes by photoinduced electron transfer
Ryuji Kojima Toshiaki Yamashita Kimiko Tanabe Tsutomu Shiragami Masahide Yasuda and Kensuke Shima pg 217; DOI: 10.1039/a605465j |
Cycloaddition vs. conjugative Michael-type addition of
2-ethoxy-3-morpholinobuta-1,3-diene with nitroolefins
Ga ![]() pg 223; DOI: 10.1039/a605345i |
1,2-Dihydroquinolin-2-one (carbostyril) anions as bidentate nucleophiles in
their reactions with aryllead triacetates: synthesis of 1-aryl- and
3-aryl-tetrahydroquinoline-2,5,8-triones
Pilar López-Alvarado Carmen Avendaño and J. Carlos Menéndez pg 229; DOI: 10.1039/a605139a |
Asymmetric reduction of 1-methylsulfonylalkan-2-ones with baker![]() Anita R. Maguire and Declan G. Lowney pg 235; DOI: 10.1039/a605132d |
Stable Cu+, Ag+ complexes of aza-bridged macrocyclic
molecules: structure and chemical properties
Hiroyuki Takemura Noriyoshi Kon Keita Tani Kô Takehara Junko Kimoto Teruo Shinmyozu and Takahiko Inazu pg 239; DOI: 10.1039/a604966d |
Chemoselective N-deprotection of tert-butyl
2-(trifluoroacetylamino) esters under PTC conditions: synthesis of
tert-butyl 2-aminocarboxylates
Domenico Albanese Francesco Corcella Dario Landini Angelamaria Maia and Michele Penso pg 247; DOI: 10.1039/a604902h |
Furan-fused 3-sulfolene as a novel building block: intermolecular
Diels–Alder reactions of
4H,6H-thieno[3,4-c]furan 5,5-dioxide
Takayoshi Suzuki Kan Kubomura and Hiroaki Takayama pg 251; DOI: 10.1039/a604600b |
Acidity effect in the regiochemical control of the alkylation of phenol
with alkenes
Giovanni Sartori Franca Bigi Raimondo Maggi and Attilio Arienti pg 257; DOI: 10.1039/a604598g |
Synthesis of chlorophyll a and ![]() Kensuke Nabeta Teruki Kawae Tatsuto Saitoh and Takahiro Kikuchi pg 261; DOI: 10.1039/a604562f |
A procedure for the preparation of cardioactive steroid precursors:
synthesis of 3![]() ![]() Lumbu Simbi and Fanie R. van Heerden pg 269; DOI: 10.1039/a604557j |
Chiral and stereoselective total synthesis of (-)-mesembranol
starting from D-glucose
Noritaka Chida Kohji Sugihara Seiji Amano and Seiichiro Ogawa pg 275; DOI: 10.1039/a604365h |
New solid-phase oligosaccharide synthesis on glycopeptides bound to a
solid phase
Hans Paulsen Axel Schleyer Nathalie Mathieux Morten Meldal and Klaus Bock pg 281; DOI: 10.1039/a604123j |
New large cage receptors. An example of selective phloroglucinol binding
Ian M. Atkinson Anthony R. Carroll Ronald J. A. Janssen Leonard F. Lindoy Owen A. Matthews and George V. Meehan pg 295; DOI: 10.1039/a604103e |
Glyceryl-ether monooxygenase [EC 1.14.16.5]. Part 9. Stereospecificity
of the oxygenase reaction
Hiroyasu Taguchi Bela Paal and Wilfred L. F. Armarego pg 303; DOI: 10.1039/a603533g |
Synthesis and reactions of lactam sulfonium salts with a sulfonio
bridgehead. Part 1.
4,4a,5,6-Tetrahydro-5-oxo-1H-thiopyrano[1,2-a]-1,4-be
nzothiazinium perchlorates
Tadashi Kataoka Yoshihide Nakamura Harutoshi Matsumoto Tetsuo Iwama Hirohito Kondo Hiroshi Shimizu Osamu Muraoka and Genzoh Tanabe pg 309; DOI: 10.1039/a603348b |
Total syntheses of (+)-asperlin, (+)-acetylphomalactone and
(5S,6S,7R,8S)-asperlin based on the
kinetic resolution of 2-furylmethanols
Zhi-Cai Yang Xiao-Bin Jiang Zhi-Min Wang and Wei-Shan Zhou pg 317; DOI: 10.1039/a603209e |
Episulfone substitution and ring-opening reactions via
![]() Allan P. Dishington Richard E. Douthwaite Andrew Mortlock Adriano B. Muccioli and Nigel S. Simpkins pg 323; DOI: 10.1039/a602846b |
Remote functionalization by tandem radical chain reactions
David Wiedenfeld pg 339; DOI: 10.1039/a600172f |
First total synthesis of carbazomycin C and D![]() Hans-Joachim Knölker and Georg Schlechtingen pg 349; DOI: 10.1039/a608351j |
Preparation, structure, derivatisation and NMR data of
cyclohexane-1,2-diacetal protected carbohydrates
Peter Grice Steven V. Ley Jörg Pietruszka Henning W. M. Priepke and Stuart L. Warriner pg 351; DOI: 10.1039/a605851e |
Synthesis of chiral intermediates of quinine alkaloids and
(+)-dihydroantirhine
Masataka Ihara Nobuaki Taniguchi and Keiichiro Fukumoto pg 365; DOI: 10.1039/a606952e |
Total synthesis of milbemycin E: synthesis of the C(11)–C(25)
fragment
Patrick G. Steel and Eric J. Thomas ![]() pg 371; DOI: 10.1039/a605892b |
Total synthesis of milbemycin E: development of a procedure for the
introduction of the 3,4-double bond and synthesis of the
C(1)–C(10) fragment
Emma R. Parmee Simon V. Mortlock Nicholas A. Stacey Eric J. Thomas and (the late) Owen S. Mills pg 381; DOI: 10.1039/a605893k |
Total synthesis of milbemycin E: resolution of the C(1)–C(10)
fragment and final assembly
Patrick G. Steel (the late) Owen S. Mills Emma R. Parmee and Eric J. Thomas pg 391; DOI: 10.1039/a605894i |
Chiral base mediated asymmetric synthesis of
tricarbonyl(![]() Richard A. Ewin Angus M. MacLeod David A. Price Nigel S. Simpkins and Alan P. Watt pg 401; DOI: 10.1039/a605812d |
Asymmetric synthesis of 5,5-disubstituted thiotetronic acids using an
allyl xanthate to dithiocarbonate rearrangement: total synthesis of
(5S)-thiolactomycin with revision of the absolute configuration
of the natural
Mark S. Chambers and Eric J. Thomas pg 417; DOI: 10.1039/a605768c |
Unusual reactions of methylsulfonyl esters: syntheses of 3![]() ![]() Michael H. Beale Huw Loaring Torren Peakman Martin Penny and Christine L. Willis pg 433; DOI: 10.1039/a605570b |
A simple method for the synthesis of 4-aryl-9-oxynaphthofuranone lignans
Kazuhiro Kobayashi Kouji Maeda Tomokazu Uneda Osamu Morikawa and Hisatoshi Konishi pg 443; DOI: 10.1039/a605288f |
Synthesis of conformationally constrained phenylalanine analogues
via 7-, 8- and 9-endo Heck cyclisations
Susan E. Gibson (née Thomas) Nathalie Guillo Richard J. Middleton Audrey Thuilliez and Matthew J. Tozer pg 447; DOI: 10.1039/a605286j |
Diazo transfer reactions of tosyl azide with carbocyclic ![]() ![]() Luisa Benati Daniele Nanni and Piero Spagnolo pg 457; DOI: 10.1039/a605240a |
Synthesis and NMR studies of key intermediates to a new class of
![]() Carla Marchioro Giorgio Pentassuglia Alcide Perboni and Daniele Donati pg 463; DOI: 10.1039/a605081f |
Fluoride ion-induced cyclization of
o-[bis(trimethylsilyl)methyl]-N-acylbenzamide
derivatives. New efficient synthesis of 2,3-differentially substituted
1(2H)-isoquinolones
Axel Couture Hélène Cornet Eric Deniau Pierre Grandclaudon and Stéphane Lebrun pg 469; DOI: 10.1039/a605077h |
Sequential and regioselective Friedel–Crafts reactions of
gem-dihalogenocyclopropanecarbonyl chlorides with benzenes for
the synthesis of 4-aryl-1-naphthol derivatives
Yoshinori Nishii and Yoo Tanabe pg 477; DOI: 10.1039/a605030a |
Reaction of 4-ethoxycarbonyl-2-phenyl-4,5-dihydrooxazol-5-one with
organolead(IV) triacetates. A route to some
![]() ![]() Mark J. Koen Jacqueline Morgan John T. Pinhey and Christopher J. Sherry pg 487; DOI: 10.1039/a604899d |
The synthesis of 3-phosphonocyclobutyl amino acid analogues of glutamic
acid via diethyl 3-oxycyclobutylphosphonate, a versatile
synthetic intermediate
Jane R. Hanrahan Paul C. Taylor and William Errington pg 493; DOI: 10.1039/a604898f |
An unexpected Mitsunobu reaction. A direct route to the
2,5-diazabicyclo[2.2.1]heptan-3-one skeleton as a ![]() ![]() Peter S. Hadfield Ron H. B. Galt Yvonne Sawyer Nicola J. Layland and Michael I. Page pg 503; DOI: 10.1039/a604564b |
Generation of homochiral aziridinium ion intermediates derived from
2,3-epoxy amines: regiospecific nucleophilic trapping with nitrogen
nucleophiles. Application in the synthesis of novel
morpholinosphingolipid analogues with potential glucosylceramide
synthase inhibitory activity
Quanying Liu Allan P. Marchington Neville Boden and Christopher M. Rayner pg 511; DOI: 10.1039/a604534k |
Stereochemistry of the methoxide induced rearrangement of an
![]() ![]() Martin J. P. Harger and Ramesh Sreedharan-Menon pg 527; DOI: 10.1039/a604093d |
Lignin model glycosides: preparation and optical resolution
Richard F. Helm Merja Toikka Kaichang Li and Gösta Brunow pg 533; DOI: 10.1039/a603786k |
Amino acids bearing nucleobases for the synthesis of novel peptide
nucleic acids
Gordon Lowe and Tirayut Vilaivan pg 539; DOI: 10.1039/a603696a |
Dipeptides bearing nucleobases for the synthesis of novel peptide
nucleic acids
Gordon Lowe and Tirayut Vilaivan pg 547; DOI: 10.1039/a603699f |
Solid-phase synthesis of novel peptide nucleic acids
Gordon Lowe and Tirayut Vilaivan pg 555; DOI: 10.1039/a603701a |
Synthesis of bicyclo[4.1.0]hept-2-enes (trinorcarenes) by photochemical
reaction of bicyclo[2.2.2]oct-5-en-2-ones
Sadamu Katayama Hajime Hiramatsu Keiichi Aoe and Masashige Yamauchi pg 561; DOI: 10.1039/a601900e |
Palladium-catalysed enantiodivergent synthesis of cis- and
trans-4-aminocyclohex-2-enols
Roberto G. P. Gatti Anna L. E. Larsson and Jan-E. Bäckvall pg 577; DOI: 10.1039/a600779a |
New approach to p-hydroxybenzylation of arenes
via a quinomethane generated in situ
from a Mannich base
Woonphil Baik Hyun Joo Lee Chang Hyun Yoo Ji Won Jung and Byeong Hyo Kim pg 587; DOI: 10.1039/a607418i |
Stereoselective synthesis of ketene telluroacetals via
hydrozirconation of acetylenic tellurides
Jin Wuk Sung Chan Pil Park Jun Mo Gil and Dong Young Oh pg 591; DOI: 10.1039/a607232a |
Additions of benzylsulfonium ylides to aldehydes and ketones: are they
under kinetic or thermodynamic control?
Varinder K. Aggarwal Simone Calamai and J. Gair Ford pg 593; DOI: 10.1039/a606925h |
Synthesis and biological testing of
pyrano[2,3-a]acridinones
Jacqueline A. Drewe and Paul W. Groundwater pg 601; DOI: 10.1039/a606689e |
Simple syntheses of L-fucopyranose and
fucosidase inhibitors utilizing the highly stereoselective methylation
of an arabinofuranoside 5-urose derivative
Shunya Takahashi and Hiroyoshi Kuzuhara pg 607; DOI: 10.1039/a606564c |
Reaction of organolead triacetates with
4-ethoxycarbonyl-2-methyl-4,5-dihydro-1,3-oxazol-5-one. The synthesis of
![]() ![]() Jacqueline Morgan John T. Pinhey and Christopher J. Sherry pg 613; DOI: 10.1039/a606309h |
2,2-Difluoro-1,3,2-oxazaborolidin-5-ones: novel approach for selective
side-chain protection of serine and threonine
Jidong Wang Yoshio Okada Wei Li Toshio Yokoi and Jintao Zhu pg 621; DOI: 10.1039/a606295d |
Synthesis of (2R)-2-bromodehydroquinic acid and
(2R)-2-fluorodehydroquinic
acid![]() Michael K. Manthey Concepción González-Bello and Chris Abell ![]() pg 625; DOI: 10.1039/a606104d |
Nitrile oxide/isoxazoline approach to higher monosaccharides: synthesis
of 7-deoxy-nonose and -decose
derivatives![]() R. Michael Paton and Anne A. Young pg 629; DOI: 10.1039/a606093e |
Facile access to 3-allyl- and
3-benzyl-![]() Hideo Tanaka Shin-ichi Sumida Kouichi Sorajo Yutaka Kameyama and Sigeru Torii pg 637; DOI: 10.1039/a606049h |
Nucleophilic introduction of fluorinated alkyl groups into aldehydes and
ketones using the corresponding alkyl halide with
samarium(II) iodide
Masato Yoshida Daiki Suzuki and Masahiko Iyoda pg 643; DOI: 10.1039/a606048j |
Preparation of N-substituted aspartic acids via
enantiospecific conjugate addition of N-nucleophiles to fumaric acids
using methylaspartase: synthetic utility and mechanistic
implications![]() M. Saeed Gulzar Mahmoud Akhtar and David Gani pg 649; DOI: 10.1039/a605996a |
Synthesis and inhibitory properties of
(1R,2R,4R,6
R)-6-O
-(2-hydroxyethyl)cyclohexane-1,2,4,6-tetraol derivatives: mechanistic
probes for the inositol monophosphatase
reaction![]() Jürgen Schulz and David Gani pg 657; DOI: 10.1039/a605998h |
Mild, effective and regioselective ring-opening of oxiranes using
several thiosilanes promoted by tetrabutylammonium fluoride as catalyst
Yoo Tanabe Kei Mori and Yoshihiro Yoshida pg 671; DOI: 10.1039/a605964c |
Pyrrolizidine alkaloid biosynthesis. Incorporation of 2-aminobutanoic
acid labelled with 13C or 2H into the senecic acid
portion of rosmarinine and senecionine
Iain R. Stirling Isabel K. A. Freer and David J. Robins pg 677; DOI: 10.1039/a605623g |
On the reaction of prop-2-enylidenetriphenylphosphorane derivatives.
Novel synthesis of the azulene ring system
Tohru Takayasu and Makoto Nitta pg 681; DOI: 10.1039/a605581h |
Catalytic conjugate addition promoted by the
copper(I)–monothiobinaphthol system. Part
2.1 Optimal ligand synthesis and initial
catalytic results
Shamsudin M. Azad Simon M. W. Bennett Stephen M. Brown Jason Green Ekkehard Sinn Chris M. Topping and Simon Woodward pg 687; DOI: 10.1039/a605620b |
A convenient synthesis of alkynylpyrazoles
Mitsuhiro Yoshimatsu Masataka Kawahigashi Eiji Honda and Tadashi Kataoka ![]() pg 695; DOI: 10.1039/a605542g |
Unusual reactions in molecules with crowded functional groups:
sulfonamide reduction under oxidizing conditions in camphor derivatives
Gabriele Wagner Rudolf Herrmann ![]() pg 701; DOI: 10.1039/a605472b |
Synthesis of 1,4-di(n-pyridyl)buta-1,3-diyne and
formation of charge-transfer complexes. X-Ray structure of
1,4-di(3-pyridyl)buta-1,3-diyne
J. Gonzalo Rodríguez Rosa Martín-Villamil Felix H. Cano and Isabel Fonseca pg 709; DOI: 10.1039/a605468d |
Synthesis of
3,4,6,7-tetrahydro-1H-5,2-benzoxathionines by
S-ylide rearrangement
Tomoko Kitano Naohiro Shirai and Yoshiro Sato pg 715; DOI: 10.1039/a605423d |
Cyclisation studies of 5-arylalkyl-1,2,3,4,5,6,7,8-octahydroisoquinolines
Philip R. Dennison Alan Gibson Alexander I. Gray and Graham L. Patrick pg 721; DOI: 10.1039/a605296g |
Dendrimeric silatrane wedges
Tim Kemmitt and William Henderson pg 729; DOI: 10.1039/a605135i |
A new approach to 1-deoxy-azasugars: asymmetric synthesis of
1-deoxymannojirimycin and 1-deoxyaltronojirimycin
Yi-Ming Xu and Wei-Shan Zhou pg 741; DOI: 10.1039/a605128f |
First examples of arylazo derivatives of
cyclooctatetraene![]() Zori V. Todres and Ghevork Ts. Hovsepyan pg 747; DOI: 10.1039/a604933h |
Syntheses of gibberellins A93 and A94, natural
products detected in wheat grain
Stuart Findlow Paul Gaskin Polly A. Harrison John R. Lenton Martin Penny and Christine L. Willis pg 751; DOI: 10.1039/a604983d |
Synthesis and biological evaluation of potential substrates for the
isolation of the strigol receptor
Jan Willem J. F. Thuring Rolf Keltjens Gerard H. L. Nefkens and Binne Zwanenburg pg 759; DOI: 10.1039/a604685a |
Synthesis and biological evaluation of strigol analogues modified in the
enol ether part
Jan Willem J. F. Thuring Angelique A. M. A. van Gaal Sander J. Hornes Margreet M. de Kok Gerard H. L. Nefkens and Binne Zwanenburg pg 767; DOI: 10.1039/a604852h |
Synthesis and stereochemistry of some new brominated spiro 1,3-dioxanes
Ion Grosu Brígida del Carmen Camacho Alfredo Toscano Gerard Plé Sorin Mager Roberto Martínez and Ruben Ramirez Gavino pg 775; DOI: 10.1039/a604734c |
Reactions of sulfonyl chlorides with silyl enol ethers catalysed by a
ruthenium(II) phosphine complex: convenient
synthesis of ![]() Nobumasa Kamigata Kumiko Udodaira and Toshio Shimizu pg 783; DOI: 10.1039/a604466b |
Formation and synthetic use of oxygen-centred radicals with
(diacetoxyiodo)arenes
Hideo Togo Takahito Muraki Yoichiro Hoshina Kentaro Yamaguchi ![]() ![]() pg 787; DOI: 10.1039/a603446b |
Dispiroketals in synthesis. Part 23.1 A new
route to (+)-D-conduritol B from
myo-inositol
Jean E. Innes Paul J. Edwards and Steven V. Ley pg 795; DOI: 10.1039/a700422b |
Copper(I)-catalysed homocoupling of
organosilicon compounds: synthesis of biaryls, dienes and diynes
Suk-Ku Kang Tae-Hyun Kim and Sung-Jae Pyun pg 797; DOI: 10.1039/a608384f |
Lithium tri-tert-butylzincate as a chemoselective
metallating reagent for functionalized organic halides
Yoshinori Kondo Michihiko Fujinami Masanobu Uchiyama and Takao Sakamoto pg 799; DOI: 10.1039/a608294g |
Synthesis of
(![]() ![]() Andrew Dinsmore Jacqueline H. Birks C. David Garner and John A. Joule pg 801; DOI: 10.1039/a607019a |
Copper-catalysed coupling of undec-10-enylmagnesium bromide with
![]() Ulrich F. Heiser and Bodo Dobner pg 809; DOI: 10.1039/a606855c |
Sulfur-controlled 5-exo selective aryl radical
cyclisation of N-vinylic 2-bromobenzamides: synthesis
of lennoxamine and chilenine
Hiroyuki Ishibashi Hirotaka Kawanami and Masazumi Ikeda pg 817; DOI: 10.1039/a606723i |
Preparation and reaction of 2-chloro-3,3-difluorocyclopropenylzinc
reagent
Yeon-Tae Jeong Ji-Hun Jung and Sam-Kwon Choi pg 823; DOI: 10.1039/a605422f |
Biosynthesis of the fungal metabolite, piliformic acid
(2-hexylidene-3-methylsuccinic acid)
Nicola C. J. E. Chesters and David O'Hagan pg 827; DOI: 10.1039/a606589i |
Acid-promoted isomerisation of 1-acceptor-1-sulfenyl-substituted
2-vinylcyclopropanes with C1–C2 bond
fission and novel 1,5-sulfenyl rearrangement
Tetsuo Iwama Harutoshi Matsumoto and Tadashi Kataoka pg 835; DOI: 10.1039/a606579a |
Syntheses of thunbergols and ![]() ![]() Peter C. Astles and Eric J. Thomas pg 845; DOI: 10.1039/a606551a |
Diastereospecific approach to ()-samin and
2,6-diaryl-3,7-dioxabicyclo[3.3.0]octane (furofuran) lignans using
the
Ireland–Claisen rearrangement of unsaturated
oxamacrolides
Hilary M. Hull née Bradley and David W Knight pg 857; DOI: 10.1039/a606545g |
Carbonylative coupling of organozinc reagents in the presence and
absence of aryl iodides: synthesis of unsymmetrical and symmetrical
ketones
Richard F. W. Jackson Debra Turner and Michael H. Block pg 865; DOI: 10.1039/a606394b |
Versatile solid-phase thiolytic reduction of azido and
N-Dts groups in the synthesis of haemoglobin
(67–76) O-glycopeptides and photoaffinity
labelled analogues to study glycan T-cell specificity
Ernst Meinjohanns Morten Meldal Teis Jensen Ole Werdelin Luisa Galli-Stampino Søren Mouritsen and Klaus Bock pg 871; DOI: 10.1039/a606725e |
Photochemical synthesis of pyrrole derivatives by desulfurization of
2,5-dihydro-1H-pyrrole-2-thiones and [2 + 2]
cycloaddition of 2,5-dihydro-1H-pyrrole-2-thiones with alkenes
Takehiko Nishio pg 885; DOI: 10.1039/a606211c |
Diacetone-glucose architecture as a chirality template. Part
9.1 Enantioselective synthesis of
(R)-mevalonolactone and
(R)-[2H9]mevalonolactone on
carbohydrate template
Masashi Kishida Noriaki Yamauchi Keiju Sawada Yuji Ohashi Tadashi Eguchi and Katsumi Kakinuma pg 891; DOI: 10.1039/a606208c |
Desilylative elimination of the quinazolinone ring from
1-(4-oxoquinazolin-3-yl)-2-silylaziridines; preparation of an N–H
aziridine in high enantiomeric excess by in situ
nucleophilic addition to the derived azirine
Robert S. Atkinson Michael P. Coogan and Ian S. T. Lochrie pg 897; DOI: 10.1039/a606092g |
1,3-Dipolar cycloaddition approach to the construction of new
bis-heterocycles from thymine as potential non-nucleoside reverse
transcriptase inhibitors
Caroline Perez Yves L. Janin David R. Adams Claude Monneret ![]() pg 901; DOI: 10.1039/a605995c |
New approach to AI-77B: stereoselective construction of a potential
precursor of the amino acid side chain
Chisato Mukai Motonori Miyakawa and Miyoji Hanaoka pg 913; DOI: 10.1039/a605901e |
Pigments of fungi. Part 43.1,2 Cardinalins
1–6, novel pyranonaphthoquinones from the fungus
Dermocybe cardinalis Horak
Malcolm S. Buchanan Melvyn Gill and Jin Yu pg 919; DOI: 10.1039/a605900g |
Exploitation of differential reactivity of the carbon–chlorine
bonds in 1,3-dichloroisoquinoline. Routes to new
N,N-chelate ligands and
1,3-disubstituted isoquinolines
Alan Ford Ekkehard Sinn and Simon Woodward pg 927; DOI: 10.1039/a605827b |
Synthesis and oxidation of chiral 2-thiazolines
(4,5-dihydro-1,3-thiazoles)
R. Alan Aitken David P. Armstrong Ronald H. B. Galt and Shaun T. E. Mesher pg 935; DOI: 10.1039/a605539g |
Tris(2,4-pentanedionato)vanadium-catalysed cyclotrimerization and
polymerization of
4-(N,N-dimethylamino)phenylethyne:
X-ray structure of
1,2,4-tris[4-(N,N
-dimethylamino)phenyl]benzene
J. Gonzalo Rodríguez Rosa Martín-Villamil and Isabel Fonseca pg 945; DOI: 10.1039/a605474i |
Synthesis of indole substituted dihydro- and tetrahydro-isoxazoles
via 1,3-dipolar cycloadditions of
C-(1-methylindol-2-yl)-N
-methylnitrone with unsaturated carbonyl derivatives and a study of
their acid-induced intramolecular
cyclizations
Elizabeth Malamidou-Xenikaki Xenophon N. Stampelos Evdoxie Coutouli-Argyropoulou Christine J. Cardin Susana Teixeira and Constantin A. Kavounis ![]() pg 949; DOI: 10.1039/a604788b |
Juncins G and H: new briarane diterpenoids of the Indian Ocean gorgonian
Junceella juncea Pallas
Ammanamanchi S. R. Anjaneyulu and Nidasanametla S. Kameswara Rao pg 959; DOI: 10.1039/a604271f |
Synthesis and crystal structure of enantiopure
N-tritylaziridin-2-ylmethanols from
L-serine and
L-threonine
Johannes G. H. Willems Marco C. Hersmis René de Gelder Jan M. M. Smits Jeannet B. Hammink F. Jan Dommerholt Lambertus Thijs and Binne Zwanenburg pg 963; DOI: 10.1039/a603801h |
Parasite glycoconjugates. Part 6.1 Chemical synthesis of
phosphorylated penta- and hepta-saccharide fragments of
Leishmania major antigenic lipophosphoglycan
Andrei V. Nikolaev Gregory M. Watt Michael A. J. Ferguson and John S. Brimacombe pg 969; DOI: 10.1039/a603800j |
Synthesis of polyfluoroalkylated bicyclic and tricyclic heterocyclic
compounds
Yan-Song Liu and Wei-Yuan Huang pg 981; DOI: 10.1039/a603071h |
Radical cyclisation with high diastereofacial selectivity: asymmetric
synthesis of ( Masataka Ihara Akira Katsumata and Keiichiro Fukumoto pg 991; DOI: 10.1039/a700834a |
Reaction of 2-alkylamino-1-azaazulenes with
N-phenylbenzylideneamine N-oxide;
one pot synthesis of the
12H-11,12,13-triazaazuleno[2,1-b
]fluorene ring system
Noritaka Abe Haruhiko Matsuda Yoshikazu Sugihara and Akikazu Kakehi pg 993; DOI: 10.1039/a700645d |
Convenient synthesis of silyl substituted butadienes; a new route to
silicon tethered intramolecular Diels–Alder reaction
precursors
Klaus Kahle Patrick J. Murphy Jonathan Scott and Roberta Tamagni pg 997; DOI: 10.1039/a700520b |
Enzymatic glycosidation in dry media under microwave
irradiation
Mirjana Gelo-Pujic Eryka Guibé-Jampel André Loupy and Antonio Trincone pg 1001; DOI: 10.1039/a700144d |
Vacuum–thermal fragmentation and ring cleavage of
1-(N-substituted-pyrrol-2-yl)-3-tosyltriazene
tetraalkylammonium salts to 4-cyano-1-azabuta-1,3-dienes
Daniele Nanni and Paolo Zanirato pg 1003; DOI: 10.1039/a606957f |
![]() ![]() Jacqueline Morgan John T. Pinhey and Bruce A. Rowe pg 1005; DOI: 10.1039/a607543f |
5-(Alk-1-enyl)-1,2,3,6-tetrahydropyridines as congeners of streptazolin
Martin Kratzel and Alexander Weigl pg 1009; DOI: 10.1039/a607309c |
D-Erythronolactone as a C4 building
unit. Part 2.1 A short and efficient synthesis
of both enantiomers of epi-muricatacin, a
diastereoisomer of the native acetogenin from Annona
muricata
Andreas Gypser Marcus Peterek and Hans-Dieter Scharf pg 1013; DOI: 10.1039/a607158i |
Synthesis of tetrahydroquinolines, hexahydrobenzoindolizines and an aryl
phosphonate linker for the generation of catalytic antibodies
Concepción González-Bello Chris Abell and Finian J. Leeper pg 1017; DOI: 10.1039/a606968a |
Synthesis of high molecular mass condensed tannin by cationic
polymerization of flavan 3,4-carbonate
Satoshi Yoneda Haruo Kawamoto and Fumiaki Nakatsubo pg 1025; DOI: 10.1039/a606783b |
Investigation of the configurational stability of lithiated phosphine
oxides using the Hoffmann test: X-ray structures of
(2S*,3S*,4R
*)-2-(N,N
-dibenzylamino)-4-diphenylphosphinoyl-1-phenylpentan-3-ol and
(2S*,4S*)-2-(N,
N
-dibenzylamino)-4-diphenylphosphinoyl-1-phenylpentan-3-one
Peter O'Brien Harold R. Powell Paul R. Raithby and Stuart Warren pg 1031; DOI: 10.1039/a606720d |
Selective mono-N-methylation of primary aromatic amines by dimethyl
carbonate over faujasite X- and Y-type zeolites
Maurizio Selva Andrea Bomben and Pietro Tundo pg 1041; DOI: 10.1039/a606684d |
New phenanthrene systems: spiro-fused tricyclic
phenanthro-1,2,4-triazolo-[4,3-d]-1,2,4-triazines and
-[3,4-d]-1,2,5-oxadiazines: ring expansions of
N-methylphenanthroazoliums
Richard N. Butler John M. McMahon Peter D. McDonald Carmel S. Pyne Simon Schambony Patrick McArdle and Desmond Cunningham pg 1047; DOI: 10.1039/a605770e |
Synthesis of functionalised fluorescent dyes and their coupling to
amines and amino acids
Mark S. J. Briggs Ian Bruce James N. Miller Christopher J. Moody Adrian C. Simmonds and Elizabeth Swann pg 1051; DOI: 10.1039/a605012c |
Synthesis, structure and stability of
E/Z-isomers of novel conjugated
enamines prepared from 9-arylmethyl- or
9-arylpropenyl-9H-carbazole with arylmethyleneanilines
Martino Paventi and Allan S. Hay pg 1059; DOI: 10.1039/a604969i |
Derivatives of L-pyrimidylalanine
Gury Zvilichovsky and Vadim Gurvich pg 1069; DOI: 10.1039/a604879j |
Conformationally locked carbocyclic nucleosides built on a
bicyclo[3.1.0]hexane template with a fixed Southern conformation.
Synthesis and antiviral activity
Abdallah Ezzitouni and Victor E. Marquez pg 1073; DOI: 10.1039/a604352f |
Expeditious synthesis of monosulfated thio-linked disaccharides
José A. Calvo-Asín Francisco G. Calvo-Flores Juan M. Exposito-López Fernando Hernández-Mateo Juan J. García-López Joaquín Isac-García Francisco Santoyo-González and Antonio Vargas-Berenguel pg 1079; DOI: 10.1039/a701345k |
Novel synthesis of the indolizidine alkaloid skeleton with appropriate
functionality and stereochemistry for use as a ![]() ![]() Elizabeth Farrant and John Mann pg 1083; DOI: 10.1039/a701193h |
Regioselective methanesulfonylation of toluene catalysed by
cation-exchanged zeolite ![]() Keith Smith Gordon M. Ewart and Kenneth R. Randles pg 1085; DOI: 10.1039/a701025g |
Synthesis of tricholomenyn A and epitricholomenyn A by a
palladium-catalysed ![]() Andrew E. Graham and Richard J. K. Taylor pg 1087; DOI: 10.1039/a700980a |
Studies towards the taxane ring system via a cascade
macrocyclisation–transannulation strategy
Stephen J. Houldsworth Gerald Pattenden David C. Pryde and Nicholas M. Thomson pg 1091; DOI: 10.1039/a700784a |
Synthesis of conjugated dienes from vinyl epoxides, vinyl acetonides and
2,5-dihydrofurans via zirconocene-mediated
deoxygenation
Sunggak Kim and Kwan Hee Kim pg 1095; DOI: 10.1039/a608593h |
An in-depth study of the biotransformation of nitriles into amides
and/or acids using Rhodococcus rhodochrous
AJ2701 Otto Meth-Cohn and Mei-Xiang Wang pg 1099; DOI: 10.1039/a607977f |
Synthetic studies relevant to biosynthetic research on vitamin
B12. Part 12.1 Modification of the
periphery of chlorins and isobacteriochlorins
James J. De Voss Finian J. Leeper and Alan R. Battersby pg 1105; DOI: 10.1039/a607852d |
Chelation-assisted nucleophilic aromatic substitution of
2-sulfonyl-substituted 1-methoxynaphthalenes by Grignard reagents:
factors determining the activating ability of the 2-sulfonyl
substituents![]() Tetsutaro Hattori Mikio Suzuki Noriyuki Tomita Ayanobu Takeda and Sotaro Miyano pg 1117; DOI: 10.1039/a607663g |
Synthesis of ![]() ![]() Steven V. Ley and Graham Meek pg 1125; DOI: 10.1039/a607376j |
A new route to ![]() Rachel Waschbüsch John Carran and Philippe Savignac pg 1135; DOI: 10.1039/a607288g |
Improved synthesis for the rodenticides, diphenacoum and brodifacoum
Pieter S. van Heerden Barend C. B. Bezuidenhoudt and Daneel Ferreira pg 1141; DOI: 10.1039/a607269k |
5-Nitrofuran-2-ylmethyl group as a potential bioreductively activated
pro-drug system
Jane M. Berry Corrine Y. Watson William J. D. Whish and Michael D. Threadgill pg 1147; DOI: 10.1039/a607202j |
Thermal fragmentation reactions of 1,4,2-dithiazines and
1,4,2,5-dithiadiazines in the presence of dienophiles: synthesis of
1,4-dithiine derivatives. X-Ray crystal structures of a 1,4,2-dithiazine
1,1-dioxide and a 1,4,2,5-dithiadiazine derivative
Martin R. Bryce Shimon Yoshida Andrei S. Batsanov and Judith A. K. Howard pg 1157; DOI: 10.1039/a606970c |
Synthesis and palladium-catalysed transformation of an annelated
barrelene
Gerald Dyker Thomas Kerl Peter G. Jones Ina Dix and Peter Bubenitschek pg 1163; DOI: 10.1039/a606857j |
Radical-mediated transannulation reactions in humulene. A new synthesis
of substituted bicyclo[6.3.0]undeca-4,9-dienes
Alexander J. Blake Amanda R. Gladwin Gerald Pattenden and Allison J. Smithies pg 1167; DOI: 10.1039/a606811a |
The synthesis of a tricyclic pyrrolopyrimidine related to
N 6-hydroxyadenine
David M. Williams Dmitry Yu. Yakovlev and Daniel M. Brown pg 1171; DOI: 10.1039/a606472h |
Synthesis of 14,17-propano analogues of estradiol
James R. Bull Clarissa Hoadley Pia G. Mountford and Lynne M. Steer pg 1179; DOI: 10.1039/a606242c |
Selective preparation of polycyclic aromatic hydrocarbons. Part
4.1 New synthetic route to anthracenes from
diphenylmethanes using Friedel–Crafts intramolecular cyclization
Takehiko Yamato Naozumi Sakaue Naoki Shinoda and Koji Matsuo pg 1193; DOI: 10.1039/a606205i |
Selective preparation of polycyclic aromatic hydrocarbons. Part
5.1 Bromination of
2,7-di-tert-butylpyrene and conversion into
pyrenoquinones and their pyrenoquinhydrones
Takehiko Yamato Masakazu Fujimoto Akira Miyazawa and Koji Matsuo pg 1201; DOI: 10.1039/a606200h |
New asymmetric route to bridged indole alkaloids: formal enantiospecific
syntheses of (-)-suaveoline, (-)-raumacline
and
(-)-N![]() Patrick D. Bailey Ian D. Collier Sean P. Hollinshead Madeleine H. Moore Keith M. Morgan David I. Smith and John M. Vernon pg 1209; DOI: 10.1039/a606081a |
Syntheses of symmetrically substituted 5-alkyl- and
5-aryl-dihydrodipyrrins and of porphyrins and bisporphyrins therefrom
David A. Lee and Kevin M. Smith pg 1215; DOI: 10.1039/a606054d |
Novel synthesis of 10-membered cyclic bis-ethers from
4-(N-alkylanilino)but-2-yn-1-ols![]() Krishna C. Majumdar Gour H. Jana and Udayan Das pg 1229; DOI: 10.1039/a606047a |
Control of the rotational barrier and spatial disposition of the
N-(2![]() Keiki Kishikawa Kazumi Yoshizaki Shigeo Kohmoto Makoto Yamamoto Kentaro Yamaguchi and Kazutoshi Yamada pg 1233; DOI: 10.1039/a605896e |
Productivity in synthesis: a mixture protocol to raise compound output
is demonstrated for asymmetric cyclopropanation of allyl alcohols
Michael D. Turnbull pg 1241; DOI: 10.1039/a605895g |
Novel class of difluorovinylphosphonate analogues of PEP
Aparecida M. Kawamoto and Malcolm M. Campbell pg 1249; DOI: 10.1039/a603094g |
Stereoselective enzymatic galactosylation of C-glucosides
Luigi Panza Pietro L. Chiappini Giovanni Russo Daniela Monti and Sergio Riva pg 1255; DOI: 10.1039/a701747b |
Anti-Markovnikov opening of trisubstituted epoxy alcohols: application
in the synthesis of 2-methyl-1,3-diols![]() Tushar K. Chakraborty and Shantanu Dutta pg 1257; DOI: 10.1039/a701536d |
Constructing the side-chain of the polyketide herbicide herboxidiene: a
protocol for the synthesis of enantiomerically enriched C-11 to C-19
fragments
Martin G. Banwell Chinh T. Bui David C. R. Hockless and Gregory W. Simpson pg 1261; DOI: 10.1039/a701360d |
Novel unsymmetrical monofunctionalized lutetium and dysprosium
bisphthalocyanines with seven crown-ether units and one hexyl
hexanoate
side-group
Didier Pernin Klaus Haberroth and Jacques Simon pg 1265; DOI: 10.1039/a701305a |
Cyclisations of benzenesulfenyl chloride adducts with conjugated
silyloxyenones: a new stereoselective reaction in the synthesis of
4,5-dihydrofuran-3(2H)-ones
Conor C. Colins Michael F. Cronin Humphrey A. Moynihan and Daniel G. McCarthy pg 1267; DOI: 10.1039/a700835j |
Photochemical behaviour of ![]() Tadashi Hasegawa Manabu Imada Yoshihiro Imase Yuko Yamazaki and Michikazu Yoshioka pg 1271; DOI: 10.1039/a700141j |
Laser-induced enantioenrichment of tartaric acid via a
multiphoton absorption process![]() Yuichi Shimizu pg 1275; DOI: 10.1039/a608453b |
Synthesis of the enantiomers of myo-inositol
1,2,4,5-tetrakisphosphate, a regioisomer of
myo-inositol 1,3,4,5-tetrakisphosphate
Stephen J. Mills and Barry V. L. Potter pg 1279; DOI: 10.1039/a608337d |
Metal-catalysed reactions of imines with ethyl diazoacetate leading to
aziridines
Kaare G. Rasmussen and Karl Anker Jørgensen pg 1287; DOI: 10.1039/a608098g |
Asymmetric addition of trimethylsilyl cyanide to aldehydes catalysed by
chiral (salen)TiIV complexes
Yuri Belokon' Massimilano Flego Nicolai Ikonnikov Margarita Moscalenko Michael North Charles Orizu Vitali Tararov and Michela Tasinazzo pg 1293; DOI: 10.1039/a608097i |
Synthesis of agonists and antagonists for central glutamate receptors by
a novel ![]() ![]() ![]() Andrew N. Bowler Andrew Dinsmore Paul M. Doyle and Douglas W. Young pg 1297; DOI: 10.1039/a608067g |
Bicyclo[3.3.1]nonanes as synthetic intermediates. Part
19.1 Asymmetric cleavage of
![]() ![]() ![]() Takefumi Momose Minoru Toshima Naoki Toyooka Yoshiro Hirai and Conrad Hans Eugster pg 1307; DOI: 10.1039/a607812e |
Bicyclo[3.3.1]nonanes as synthetic intermediates. Part
20.1 Asymmetric synthesis of the indolizidine
alkaloids monomorine I and indolizidine 223AB
Takefumi Momose Minoru Toshima Sumie Seki Yayoi Koike Naoki Toyooka and Yoshiro Hirai pg 1315; DOI: 10.1039/a607981d |
Simple preparation of fused
pyrrolo[2,3-b]pyrrolidinones and
pyrrolo[2,3-c]pyridazinones![]() Yoshinari Okamoto Yumiko Kaneda Tetsuo Yamasaki Tadashi Okawara and Mitsuru Furukawa pg 1323; DOI: 10.1039/a607816h |
In search of open-chain 1,3-stereocontrol
Asun Barbero David C. Blakemore Ian Fleming and Robert N. Wesley pg 1329; DOI: 10.1039/a607545b |
A new chiral synthesis of bullfrog bile sterol 5![]() Don W. Harney and Theodore A. Macrides pg 1353; DOI: 10.1039/a607850h |
Alkaline earth metal-sensing anthracene fluorophore-hosts
Satoru Iwata Hideo Matsuoka and Kiyoshi Tanaka pg 1357; DOI: 10.1039/a607688b |
Acylation of in situ generated trimethylsilyl
diethylphosphonoacetate using magnesium chloride–triethylamine: a
practical synthesis of ![]() Dae Young Kim Myeon Sik Kong and Kilsung Lee pg 1361; DOI: 10.1039/a607683a |
Internally quenched fluorogenic, ![]() Seema Mehta Morten Meldal Vito Ferro Jens Ø. Duus and Klaus Bock pg 1365; DOI: 10.1039/a607624f |
o-Nitroaniline derivatives. Part
14.1,2 Cyclisations leading to benzimidazole
N-oxides, N-hydroxybenzimidazolones
and N-hydroxyquinoxaline-2,3-diones: a mechanistic
borderline
Pamela A. Collins Cafiero Colin S. French Michael D. McFarlane Raymond K. Mackie and David M. Smith pg 1375; DOI: 10.1039/a607378f |
Synthesis based on cyclohexadienes. Part 22.1
Formal syntheses of patchouli alcohol and norpatchoulenol
Krishna P. Kaliappan and G. S. R. Subba Rao pg 1385; DOI: 10.1039/a607286k |
Highly selective conversion of hydroxylated biaryls to dibenzofuran
derivatives over zeolite catalyst
Attilio Arienti Franca Bigi Raimondo Maggi Pietro Moggi Massimo Rastelli Giovanni Sartori and Alessandra Trerè pg 1391; DOI: 10.1039/a607282h |
2,2![]() ![]() Joseph Frey and Zvi Rappoport pg 1395; DOI: 10.1039/a607222d |
Synthesis of the monomeric unit of ![]() Margaret A. Brimble Letecia J. Duncalf and Sara J. Phythian pg 1399; DOI: 10.1039/a606765d |
Retinoids and related compounds. Part 19.1
Syntheses of 9E- and 9Z-locked
retinoic acid analogues and their transcriptional activities as ligands
for retinoic acid receptors and retinoid X receptors
Yuko Katsuta Yukiko Aoyama Hisa Osone Akimori Wada and Masayoshi Ito pg 1405; DOI: 10.1039/a606719k |
Palladium-catalysed asymmetric allylic substitution: synthesis of
![]() ![]() Justin F. Bower Roshan Jumnah Andrew C. Williams and Jonathan M. J. Williams pg 1411; DOI: 10.1039/a606586d |
Synthesis of the aromatic unit of calicheamicin
![]() Yong-Zhou Hu and Derrick L. J. Clive pg 1421; DOI: 10.1039/a605837j |
Unexpected stereoselectivity in the Weiss–Cook condensation of
dimethyl 1,3-acetonedicarboxylate with pentane-2,3-dione
Richard Vaughan Williams Vijay R. Gadgil Ashwani Vij James M. Cook Greg Kubiak and Qi Huang pg 1425; DOI: 10.1039/a605817e |
Glycosylation of Fmoc amino acids: preparation of mono- and
di-glycosylated derivatives and their incorporation into Arg-Gly-Asp
(RGD)-containing glycopeptides
Hiran Vegad Charles J. Gray Peter J. Somers and Anand S. Dutta pg 1429; DOI: 10.1039/a604372k |
Synthesis and reactions of 3,3![]() Chitoshi Kitamura and Yoshiro Yamashita pg 1443; DOI: 10.1039/a700154a |
A new synthetic method for the preparation of amino sugars through an
allyl cyanate-to-isocyanate rearrangement
Yoshiyasu Ichikawa Masafumi Osada Ikuko I. Ohtani and Minoru Isobe pg 1449; DOI: 10.1039/a700142h |
Reactions involving fluoride ion. Part 42.1
Heterocyclic compounds from perfluoro-3,4-dimethylhexa-2,4-diene
Richard D. Chambers William K. Gray Steven J. Mullins and Stewart R. Korn pg 1457; DOI: 10.1039/a608584i |
The in situ generation of alk-1-ynyllead triacetates
from terminal acetylenes by zinc–lead exchange and crystal
structure of
2,4,7,9,13-pentamethyl-9-phenylethynyl-7,10-ethenospiro[5.5]undeca-1,4-
diene-3,8-dione
Christopher J. Parkinson Trevor W. Hambley and John T. Pinhey pg 1465; DOI: 10.1039/a608582b |
The synthesis of alkylated or acylated nitroarene cyclopentadienyliron
complexes: an alternative approach to the synthesis of arylated
alkanoates
Alaa S. Abd-El-Aziz Waleed Boraie Najeeb Al-Salem Salwa A. Sadek and Karen M. Epp pg 1469; DOI: 10.1039/a608578d |
Preparation of ![]() Iain Coldham Stuart Holman and Maria M. S. Lang-Anderson pg 1481; DOI: 10.1039/a608576h |
Reactions of
2-methyl-4H-pyrido[2,3-d][3,1]oxazin-4-one with active
methylene compounds: a new efficient route to 3-substituted
4-hydroxy-1,8-naphthyridin-2(1H)-ones
Vassiliki Delieza Anastasia Detsi Vassilios Bardakos and Olga Igglessi-Markopoulou pg 1487; DOI: 10.1039/a608509a |
Mechanism of the Stevens rearrangement of ammonium ylides
Yasuhiro Maeda and Yoshiro Sato pg 1491; DOI: 10.1039/a608492c |
Synthesis of pendant polyaminopolycarboxylic acid crown ethers:
potential ligands for MRI contrasting agents
B. Lakshmi A. Prabhavathi Devi and Madhavarao Nagarajan pg 1495; DOI: 10.1039/a608452d |
Building units for N-backbone cyclic peptides. Part 4.1
Synthesis of protected N![]() Gal Bitan Dan Muller Ron Kasher Evgenia V. Gluhov and Chaim Gilon pg 1501; DOI: 10.1039/a608389g |
Aryltricyclospirodienones; novel steroid mimics as inhibitors of
aromatase
David Hobbs-Mallyon Warren Li and Donald A. Whiting pg 1511; DOI: 10.1039/a608338b |
Diastereoselective acyclic aza-[2,3] Wittig sigmatropic
rearrangements
James C. Anderson Stephen C. Smith and Martin E. Swarbrick pg 1517; DOI: 10.1039/a608226b |
Secondary mould metabolites: Part 53.1
Transformation of the protoilludane sesquiterpene tsugicoline A into a
sterpurane derivative and its microbiological reduction
Alberto Arnone Cristiana De Gregorio Gianluca Nasini and Orso Vajna De Pava pg 1523; DOI: 10.1039/a608174f |
Enantioselective synthesis of ![]() Tsutomu Yokomatsu Takehiro Yamagishi and Shiroshi Shibuya pg 1527; DOI: 10.1039/a608161d |
Novel photochemical behaviour of the oximes and hydrazones of
![]() ![]() Diego Armesto Ana Ramos Maria J. Ortiz William M. Horspool Maria J. Mancheño Olga Caballero and Elena P. Mayoral pg 1535; DOI: 10.1039/a607435i |
A radio-iodinated abscisic acid photoaffinity probe
Andrew D. Kohler Michael H. Beale Ruth Rollason D. H. Paul Barratt Mervyn J. Lewis R. M. Van der Meulen and Mei Wang pg 1543; DOI: 10.1039/a607307g |
Synthesis of functionalised indolines by radical-polar crossover
reactions
John A. Murphy Faiza Rasheed Stéphane Gastaldi T. Ravishanker and Norman Lewis pg 1549; DOI: 10.1039/a607060d |
Nitration of ![]() ![]() Stuart A. Hewlins John A. Murphy Jian Lin David E. Hibbs and Michael B. Hursthouse pg 1559; DOI: 10.1039/a607170h |
Novel synthesis of degradation products of carotenoids,
megastigmatrienone analogues and blumenol-A
Nobuhiko Ito Takeaki Etoh Hisahiro Hagiwara and Michiharu Kato pg 1571; DOI: 10.1039/a607028k |
Asymmetric 1,3-dipolar cycloaddition of optically active
trifluoromethylated ![]() ![]() Hiroyasu Tsuge Takashi Okano Shoji Eguchi and Hiroshi Kimoto pg 1581; DOI: 10.1039/a606890a |
Harzianin HB I, an 11-residue peptaibol from Trichoderma
harzianum: isolation, sequence, solution synthesis and membrane
activity
Isabelle Augeven-Bour Sylvie Rebuffat Catherine Auvin Christophe Goulard Yann Prigent and Bernard Bodo pg 1587; DOI: 10.1039/a605629f |
Efficient cyclopropanation of C60 starting from malonates
Xavier Camps and Andreas Hirsch pg 1595; DOI: 10.1039/a702055d |
Synthesis of (difluoromethyl)phosphonate azasugars designed as
inhibitors for glycosyl transferases
Jean-Bernard Behr Claude Mvondo Evina Nga Phung and Georges Guillerm pg 1597; DOI: 10.1039/a700800g |
Short path syntheses of ![]() Yuxiang Dong Karl Griesbaum and Kevin J. McCullough pg 1601; DOI: 10.1039/a700989e |
Gas-phase pyrolysis of 1-(2-azidophenyl)imidazole
Alexander J. Blake Bernard A. J. Clark Hamish McNab and Craig C. Sommerville pg 1605; DOI: 10.1039/a700457e |
Unexpected formation of highly stabilized
tetrakis-(2-alkoxyphenyl)bismuthonium salts in the oxidation of
tris-(2-alkoxyphenyl)bismuthanes with iodosylbenzene
Hitomi Suzuki Tohru Ikegami and Nagao Azuma pg 1609; DOI: 10.1039/a700379j |
Reaction of furans with trithiazyl trichloride: a new synthesis of
isothiazoles
Xiao-Lan Duan Ross Perrins and Charles W. Rees pg 1617; DOI: 10.1039/a700358g |
Conversion of carbonimidodithioates to carbamates
Mariappan Anbazhagan T. Indrasena Reddy and Srinivasachari Rajappa pg 1623; DOI: 10.1039/a700166e |
Synthesis of homoallylic (but-3-enylic) alcohols from aldehydes with
allylic chlorides, tin(II) chloride and potassium iodide in
water
Didier Houllemare Francis Outurquin and Claude Paulmier pg 1629; DOI: 10.1039/a608487g |
Synthesis of methyl secolonitoside
Richard T. Brown Stephen P. Mayalarp and Joanne Watts pg 1633; DOI: 10.1039/a608247e |
![]() David Soullez Gérard Plé and Lucette Duhamel pg 1639; DOI: 10.1039/a608187h |
Chemistry of the mycalamides: antiviral and antitumour compounds from a
New Zealand marine sponge. Part 6.1–3 The
synthesis and testing of analogues of the C(7)–C(10) fragment
Andrew D. Abell John W. Blunt Glenn J. Foulds and Murray H. G. Munro pg 1647; DOI: 10.1039/a608168a |
Chemistry and X-ray crystallographic structure of N-protected
(5-oxo-1,3-oxazolidin-4-yl)acetic acids: versatile intermediates in the
synthesis of peptidomimetics
Andrew D. Abell Ross A. Edwards and Mark D. Oldham pg 1655; DOI: 10.1039/a608165g |
Preparation and biological activity of tricyclic non-steroidal
inhibitors of human steroid 5![]() Andrew D. Abell Martin Brandt Mark A. Levy ![]() ![]() pg 1663; DOI: 10.1039/a608169j |
Furan-2(3H)- and -2(5H)-ones. Part
7.1 Photochemical behaviour of tetrahydro- and
hexahydro-isobenzofuran-1-one systems: a mechanistic and exploratory
study
Osamu Muraoka Genzoh Tanabe and Yuko Igaki pg 1669; DOI: 10.1039/a608122c |
Alkylation of chiral
2-(aminomethyl)oxazolines![]() Marc Le Bail David J. Aitken Fabrice Vergne and Henri-Philippe Husson pg 1681; DOI: 10.1039/a608030h |
Synthesis and Diels–Alder reactions of
2-acetamido-3-phenylthiobuta-1,3-diene and its derivatives
Shang-Shing P. Chou Tahsin J. Chow Chien-Hung Hsu Chengda Yang Shu-Hua Long and Chih-Da Lin pg 1691; DOI: 10.1039/a607817f |
Indolisation of 1-decalone and the reactions of the products with oxygen
and with nucleophiles
David W. Brown Mary F. Mahon Aleyamma Ninan and Malcolm Sainsbury pg 1699; DOI: 10.1039/a607577k |
Total synthesis of ()-furoscrobiculin B
Maki Seki Toshihiro Sakamoto Hiroshi Suemune and Ken Kanematsu pg 1707; DOI: 10.1039/a607164c |
Bacterial dioxygenase-catalysed dihydroxylation and chemical resolution
routes to enantiopure cis-dihydrodiols of chrysene
Derek R. Boyd Narain D. Sharma Rajiv Agarwal Sol M. Resnick Mark J. Schocken David T. Gibson Jane M. Sayer Haruhiko Yagi and Donald M. Jerina pg 1715; DOI: 10.1039/a606686k |
Synthesis and conformational studies of
tetrahydroxy[3.1.3.1]metacyclophanes and electrophilic aromatic
substitution of their tetramethoxy derivatives
Takehiko Yamato Yoshiyuki Saruwatari and Masashi Yasumatsu pg 1725; DOI: 10.1039/a606358f |
Synthesis and conformational studies of regio- and conformational
isomers derived by O-alkylation of
tetrahydroxy[3.1.3.1]metacyclophane![]() Takehiko Yamato Yoshiyuki Saruwatari and Masashi Yasumatsu pg 1731; DOI: 10.1039/a606354c |
Asymmetric hydrolysis of pro-chiral 3,3-disubstituted
2,4-diacetoxycyclohexa-1,4-dienes
Philippe Renouf Jean-Marie Poirier and Pierre Duhamel pg 1739; DOI: 10.1039/a606001c |
Preparation of optically active photopyridone by lipase-catalysed
asymmetric resolution![]() Hiroshi Hongo Kazuto Iwasa Chizuko Kabuto Hisao Matsuzaki and Hiroto Nakano pg 1747; DOI: 10.1039/a605698i |
Synthesis of ()-trans-cyclohexa-3,5-diene-1,2-diol
derivatives from myo-inositol
Hari Babu Mereyala and Madhavi Pannala pg 1755; DOI: 10.1039/a605576a |
Design of new chiral tetraol host compounds,
trans-1,4-bis[3-(o-chlorophenyl)-3-hydroxy-3-
phenylprop-1-ynyl]-1,4-dihydroxycyclohexa-2,5-diene and its
tetrahalogeno derivatives
Fumio Toda and Tomonori Shinyama pg 1759; DOI: 10.1039/a701874f |
Enantioselective Pummerer-type rearrangement by reaction of
O-silylated ketene acetal with enantiopure
![]() Yasuyuki Kita Norio Shibata Seiji Fukui Masahiko Bando and Shigekazu Fujita pg 1763; DOI: 10.1039/a702020a |
Cleavage of (octaethyl-2,3-dihydroxychlorinato)nickel(II) to
give the novel 2,3-dioxo-2,3-secochlorin system
Keith R. Adams Raymond Bonnett Philip J. Burke Antonio Salgado and María Asunción Vallés pg 1769; DOI: 10.1039/a701152k |
Retinoids and related compounds. Part 20.1 Synthesis of
(11Z)-8,18-ethanoretinal and a conformational study of the
rhodopsin chromophore
Akimori Wada Miho Sakai Yasushi Imamoto Yoshinori Shichida Masashige Yamauchi and Masayoshi Ito pg 1773; DOI: 10.1039/a700796e |
Regio- and stereo-chemical outcomes in the nucleophilic ring cleavage
reactions of mono-epoxides derived from
cis-1,2-dihydrocatechols
Martin G. Banwell Najiba Haddad Tomas Hudlicky Thomas C. Nugent Maureen F. Mackay and Sharon L. Richards pg 1779; DOI: 10.1039/a700733g |
Enantioselective synthesis of 2-isocephem and 2-isooxacephem antibiotics
Hajime Nitta Ikuo Ueda and Minoru Hatanaka pg 1793; DOI: 10.1039/a700650k |
Preparation and pyrolysis of 1-(pyrazol-5-yl)-1,2,3-triazoles and
related compounds![]() David Clarke Richard W. Mares and Hamish McNab pg 1799; DOI: 10.1039/a700421d |
Enantiospecific synthesis of (-)-5-epi-shikimic
acid and (-)-shikimic acid
Shende Jiang Kevin J. McCullough Boualem Mekki Gurdial Singh and Richard H. Wightman pg 1805; DOI: 10.1039/a700389g |
Chemistry of zamoranic acid. Part 10. Homochiral
hemisynthesis of pereniporin A
Julio G. Urones David Díez Patricio M. Gómez Isidro S. Marcos Pilar Basabe and Rosalina F. Moro pg 1815; DOI: 10.1039/a700377c |
Synthesis and conjugate additions of
2,3,4,9-tetrahydro-1H-xanthene-1,9-diones
Christopher D. Gabbutt John D. Hepworth Michael W. J. Urquhart and Luis Millan Vazquez de Miguel pg 1819; DOI: 10.1039/a700375g |
Synthesis of oligodeoxynucleotides containing
6-N-([13C]methyl)adenine and
2-N-([13C]methyl)guanine
Mechtild Hofmann Montse Acedo Patricia Fagan David Wemmer Ramon Eritja and Antonio R. Díaz pg 1825; DOI: 10.1039/a700366h |
Cleavage and reactions of some NH-BOC protected 1-aminopyrroles: a new
one-pot route to pyrrolo[1,2-b][1,2,4]triazines together with
spectroscopic and X-ray studies
Orazio A. Attanasi Lucia De Crescentini Elisabetta Foresti Giuseppe Gatti Raffaello Giorgi Francesca R. Perrulli and Stefania Santeusanio pg 1829; DOI: 10.1039/a700355b |
Stereoselective synthesis of (-)-metasequoic acid B
Antonio Abad Consuelo Agulló Manuel Arnó Angel Cantín Ana C. Cuñat Benjamín Meseguer and Ramón J. Zaragozá pg 1837; DOI: 10.1039/a700354d |
Phospholipase-A2-mediated stereoselective synthesis of
(R)-1-O-alkylglycero-3-phosphate and alkyl-acyl
analogues: application for synthesis of radiolabelled biosynthetic
precursors of cell surface glycoconjugates of Leishmania
donovani
Parmeshwari Sahai and Ram A. Vishwakarma pg 1845; DOI: 10.1039/a700353f |
Photochemical reactions of thiobenzamides bearing an allylic substituent
on the nitrogen atom: double-bond migration via tandem 1,4- and
1,6-hydrogen transfer
Hiromu Aoyama pg 1851; DOI: 10.1039/a700247e |
Efficient synthesis of
O-(2-acetamido-2-deoxy-![]() ![]() Uttam K. Saha and Richard R. Schmidt pg 1855; DOI: 10.1039/a700210f |
[4 + 2]Cycloaddition of indole derivatives with
bismaleimides: a route to new biscarbazoles
Ulf Pindur Eugenia Gonzalez and Farokh Mehrabani pg 1861; DOI: 10.1039/a608580f |
Asymmetric hydrogenation of acrylic acid derivatives by novel chiral
rhodium–phosphinediamine complex catalysts by selective ligation
between two amino units of the ligand and electrostatic interaction
Issaku Yamada Munetaka Ohkouchi Motowo Yamaguchi and Takamichi Yamagishi pg 1869; DOI: 10.1039/a608228i |
Regioselective total synthesis of edulane and its angular analogue
Kandasamy Subburaj Modachur G. Murugesh and Girish K. Trivedi pg 1875; DOI: 10.1039/a608227k |
Toluene dioxygenase-catalysed oxidation route to angular
cis-monohydrodiols and other bioproducts from bacterial
metabolism of 1,2-dihydrobenzocyclobutene and derivatives
Derek R. Boyd Narain D. Sharma Timothy A. Evans Melanie Groocock John F. Malone Paul J. Stevenson and Howard Dalton pg 1879; DOI: 10.1039/a608071e |
Synthesis of 2-substituted 2![]() Christine Edwards Gernot Boche Thomas Steinbrecher and Susanne Scheer pg 1887; DOI: 10.1039/a604559f |
19-Hydroxy-5![]() John F. Templeton Yangzhi Ling Weiyang Lin Helena Majgier-Baranowska and Kirk Marat pg 1895; DOI: 10.1039/a604405k |
Polymer supported perruthenate (PSP): a new oxidant for clean organic
synthesis
Berthold Hinzen and Steven V. Ley pg 1907; DOI: 10.1039/a703461j |
TiCl4-promoted cross-coupling reaction of dialkyl
3,3,3-trifluoropropyl acetals for the preparation of
CF3-containing functionalized compounds
Feng Hong and Chang-Ming Hu pg 1909; DOI: 10.1039/a702402i |
Convergent, enantioselective synthesis of the novel furanoditerpene
(+)-taonianone through facially selective chiral
olefin–ketene [2+2] cycloaddition
Alice Kanazawa Philippe Delair Mehrnaz Pourashraf and Andrew E. Greene pg 1911; DOI: 10.1039/a701629h |
Angular trifluoromethyl group. Part 6.1 Studies in the
series of 19,19,19-trifluoroandrostenedione![]() Jean-Claude Blazejewski Jean Guilhem and Frédéric Le Guyader pg 1913; DOI: 10.1039/a701876b |
Metal cation-exchanged montmorillonite
(Mn+-mont)-catalysed aromatic alkylation with
aldehydes and ketones
Jun-ichi Tateiwa Ei Hayama Takahiro Nishimura and Sakae Uemura pg 1923; DOI: 10.1039/a701744h |
Intramolecular Diels–Alder additions to 2-benzopyran-3-ones;
anti-selectivity induced by the phenylsulfonyl
group![]() Edward J. Bush David W. Jones and Tracie C. L. M. Ryder pg 1929; DOI: 10.1039/a701589e |
Synthesis of 1,2,4-dioxazolidine derivatives by the ozonolysis of
indenes in the presence of primary amines
Yoshihiro Ushigoe Syuzo Satake Araki Masuyama Masatomo Nojima and Kevin J. McCullough pg 1939; DOI: 10.1039/a701572k |
Oligomeric flavanoids. Part 26. Structure and
synthesis of the first profisetinidins with epifisetinidol constituent
units
Petrus J. Steynberg Jan P. Steynberg E. Vincent Brandt Daneel Ferreira and Richard W. Hemingway pg 1943; DOI: 10.1039/a701334e |
Automated synthesis of branched oligodeoxynucleotide analogues using
arabino-uridine as branching nucleotide
Michael Meldgaard Nanna K. Nielsen Murray Bremner Ole S. Pedersen Carl Erik Olsen and Jesper Wengel pg 1951; DOI: 10.1039/a701228d |
Synthesis of 3,4![]() ![]() ![]() ![]() ![]() ![]() Luciano Antolini Francesca Goldoni Dario Iarossi Adele Mucci and Luisa Schenetti pg 1957; DOI: 10.1039/a700811b |
Synthesis of ![]() ![]() ![]() ![]() ![]() Christine Wedler Katharina Kleiner Egon Gründemann and Hans Schick pg 1963; DOI: 10.1039/a700805h |
Convenient and stereospecific homologation of
N-fluorenylmethoxycarbonyl-![]() ![]() Antonella Leggio Angelo Liguori Antonio Procopio and Giovanni Sindona pg 1969; DOI: 10.1039/a700731k |
Synthesis of neoglycoproteins containing
L-glycero-![]() ![]() ![]() ![]() Harald Sekljic Norbert Wimmer Andreas Hofinger Helmut Brade and Paul Kosma pg 1973; DOI: 10.1039/a700497d |
Three component aminoalkylation of aldehydes by functionalized
organozinc compounds promoted by lithium perchlorate (LiClO4)
Mohammad R. Saidi Hamid R. Khalaji and Junes Ipaktschi pg 1983; DOI: 10.1039/a700371d |
Silyl enol ethers as new protecting groups for alkyl
4-halo-3-oxobutanoates; the preparation of pure
(3-alkoxycarbonyl-2-oxopropyl)triphenylphosphonium salts
Cornelis M. Moorhoff pg 1987; DOI: 10.1039/a700241f |
Molecular engineering. Part 2.1 Influence of side-chain
substituents in lariat-type upper-rim calix[4]crowns on their binding
properties and the reversal of these
Hyejae Ihm Hyunjun Kim and Kyungsoo Paek pg 1997; DOI: 10.1039/a700165g |
Bicyclo[3.3.1]nonanes as synthetic intermediates. Part
21.1 Enantiodivergent synthesis of the
cis,cis 2,6-disubstituted piperidin-3-ol chiral
building block for alkaloid synthesis
Takefumi Momose Naoki Toyooka and Makoto Jin pg 2005; DOI: 10.1039/a608490g |
Synthesis and characterization of 2-methoxy-2H-azepines: the
first isolation of 2-azanorcaradiene, the valence isomer of
3H-azepine
Kyosuke Satake Yuko Tawada Hideki Okamoto and Masaru Kimura pg 2015; DOI: 10.1039/a703709k |
First synthesis of sulfines by direct oxidation of
xanthates![]() Eddie Marrière David Chevrie and Patrick Metzner pg 2019; DOI: 10.1039/a703706f |
New and efficient approach to the synthesis of pentacoordinate
spirobicyclic phosphoranes
Hua Fu Guang-Zhong Tu Zhao-Long Li Yu-Fen Zhao and Ri-Qing Zhang pg 2021; DOI: 10.1039/a702813j |
Direct preparation of diacetals from 1,2-diketones and their use as
1,2-diol protecting groups
Achim Hense Steven V. Ley Helen M. I. Osborn Dafydd R. Owen Jean-François Poisson Stuart L. Warriner and Kieron E. Wesson pg 2023; DOI: 10.1039/a702497e |
Evidence for oxacarbenium ion intermediates in the Lewis acid promoted
cleavage of spirocyclic dioxanes
Lee A. Newitt and Patrick G. Steel pg 2033; DOI: 10.1039/a701764b |
Synthesis of 19-hydroxy-1![]() John F. Templeton Weiyang Lin Yangzhi Ling Helena Majgier-Baranowska and Kirk Marat pg 2037; DOI: 10.1039/a701570d |
Biomimetic synthesis of a peptide antibiotic, gratisin
Makoto Tamaki Seiji Komiya Sadatoshi Akabori and Ichiro Muramatsu pg 2045; DOI: 10.1039/a701537b |
Synthesis of oligodeoxynucleotides containing 5-aminouracil and its
N-acetyl derivative
Elisenda Ferrer Gitte Neubauer Matthias Mann and Ramon Eritja pg 2051; DOI: 10.1039/a701371j |
Synthesis of indoles and quinolones by sequential Wittig and Heck
reactions
Elliot J. Latham and Stephen P. Stanforth pg 2059; DOI: 10.1039/a701282i |
In vitro biosynthesis of cadinanes by cell-free extracts of
cultured cells of Heteroscyphus planus
Kensuke Nabeta Masaru Fujita Kaori Komuro Kinya Katayama and Toshihide Takasawa pg 2065; DOI: 10.1039/a701145h |
Thermolysis and CoII-tetraphenylporphyrin-catalysed
decomposition of substituted cycloheptatriene endoperoxides: a new
synthetic approach to substituted dihydrooxepines
M. Emin Sengül and Metin Balci pg 2071; DOI: 10.1039/a701105i |
1-Substituted 2![]() Lorenzo De Napoli Anna Messere Daniela Montesarchio Gennaro Piccialli and Michela Varra pg 2079; DOI: 10.1039/a700987i |
Design, synthesis and pharmacological test of a quinoline based,
nonpeptidic analogue of neurotensin(8–13)
Feng Hong Yuan-Ping Pang Bernadette Cusack and Elliott Richelson pg 2083; DOI: 10.1039/a700894e |
Homoproline homologation by enolate Claisen rearrangement or
direct allylation: syntheses of (-)-trachelanthamidine,
(-)-isoretronecanol and
()-turneforcidine
David W. Knight Andrew C. Share and Peter T. Gallagher pg 2089; DOI: 10.1039/a700792b |
Haem d1: stereoselective synthesis of the reduced
form of its parent macrocycle using the original coupling strategy
Christopher J. Aucken Finian J. Leeper and Alan R. Battersby pg 2099; DOI: 10.1039/a700652g |
Haem d1: development of a new coupling procedure
leading to the synthesis of isobacteriochlorins![]() Richard L. Mackman Jason Micklefield Michael H. Block Finian J. Leeper and Alan R. Battersby pg 2111; DOI: 10.1039/a700654c |
Haem d1: stereoselective synthesis of the macrocycle
to establish its absolute configuration as
2R,7R![]() Jason Micklefield Marion Beckmann Richard L. Mackman Michael H. Block Finian J. Leeper and Alan R. Battersby pg 2123; DOI: 10.1039/a700655a |
Synthesis and pyrolytic behaviour of thiazolidin-2-one 1,1-dioxides
R. Alan Aitken David P. Armstrong Ronald H. B. Galt and Shaun T. E. Mesher pg 2139; DOI: 10.1039/a700521k |
Isolation and sequence analysis of the peptide antibiotics trichorzins
PA from Trichoderma harzianum
Delphine Duval Sylvie Rebuffat Christophe Goulard Yann Prigent Michel Becchi and Bernard Bodo pg 2147; DOI: 10.1039/a700244k |
Ring-opening reactions of functionalized bicyclo[2.2.0]hexanes
M. Liliana Graziano M. Rosaria Iesce Flavio Cermola and Giuseppina Ialongo pg 2155; DOI: 10.1039/a607507j |
Chiral base-mediated asymmetric functionalisation of
tricarbonylchromium(0) complexes of benzyl sulfides
Susan E. Gibson Peter Ham Gary R. Jefferson and Mark H. Smith pg 2161; DOI: 10.1039/a704252c |
Synthesis of new trialkylsilylmethyloxazinones via
intramolecular trapping of ![]() Sylvie Brocherieux-Lanoy Hamid Dhimane Jean-Christophe Poupon Corinne Vanucci and Gérard Lhommet pg 2163; DOI: 10.1039/a703902f |
Unusual condensation of 2-(2-dimethylaminovinyl)-1-benzopyran-4-one with
dimethyl acetylenedicarboxylate: formation of
2,3-bis(methoxycarbonyl)xanthen-9-one
Chandra Kanta Ghosh Samita Bhattacharyya and Amarendra Patra pg 2167; DOI: 10.1039/a703495d |
Metal cation-exchanged
montmorillonite(Mn+-Mont)-catalysed
carbonyl-ene reactions
Jun-ichi Tateiwa Akihiro Kimura Masaaki Takasuka and Sakae Uemura pg 2169; DOI: 10.1039/a702906c |
An expeditious synthesis of chaetomellic anhydrides A and B, and
analogues
Stéphane Poigny Michèle Guyot and Mohammad Samadi pg 2175; DOI: 10.1039/a702668d |
Total synthesis of (-)-slaframine from
(2R,3S)-3-hydroxyproline
David W. Knight and A. William Sibley pg 2179; DOI: 10.1039/a701878i |
Synthesis and some reactions of
N-amino-2-methoxy-1-azaazulenium salt: leading to
3,3a-diazacyclopent[a]azulene and
2a,3-diazabenz[cd![]() Abe Noritaka Kunihiko Odagiri and Akikazu Kakehi pg 2189; DOI: 10.1039/a701793f |
Synthesis of pyrrolizin-3-ones by flash vacuum pyrolysis of
pyrrol-2-ylmethylidene Meldrum![]() Shirley E. Campbell Murray C. Comer Paul A. Derbyshire Xavier L. M. Despinoy Hamish McNab Roderick Morrison Craig C. Sommerville and Craig Thornley pg 2195; DOI: 10.1039/a701749i |
New synthetic routes to pyrrolo-[1,2-a]- and
-[1,2-c]-imidazol-5-ones by flash vacuum pyrolysis
Hamish McNab and Craig Thornley pg 2203; DOI: 10.1039/a701751k |
Synthesis and structural characteristics of novel
5H-thiazolo[2,3-d][1,5]benzothiazepine derivatives
Giuseppe Bruno Alba Chimirri Rosaria Gitto Silvana Grasso Francesco Nicolò Rosario Scopelliti and Maria Zappalà pg 2211; DOI: 10.1039/a701539i |
Abnormal products in the Bischler–Napieralski isoquinoline
synthesis
Satoshi Doi Naohiro Shirai and Yoshiro Sato pg 2217; DOI: 10.1039/a701332i |
Approaches to pseudopeptidic ergopeptines. Part 3.1
Consequences of the incorporation of an
![]() Anna Calcagni Gino Lucente Grazia Luisi Francesco Pinnen Domenico Rossi and Enrico Gavuzzo pg 2223; DOI: 10.1039/a701230f |
Approaches to 1,1-disubstituted cinnolin-3-ylio oxides: synthesis and
reactivity of a new class of heterocyclic betaines
Vicente J. Arán Juan L. Asensio José Molina Pilar Muñoz José R. Ruiz and Manfred Stud pg 2229; DOI: 10.1039/a701103b |
Synthesis and biological activity of side-chain analogues of ecdysone
and 20-hydroxyecdysone
Patrick G. Roussel Vladimir Sik Nicholas J. Turner and Laurence N. Dinan pg 2237; DOI: 10.1039/a700986k |
Further reactions of furans with trithiazyl trichloride; mechanistic
considerations
Charles W. Rees and Tai-Yuen Yue pg 2247; DOI: 10.1039/a700488e |
Synthesis of enantiomerically pure (1R,2R)- and
(1S,2S)-2-alkyl-1-phenylsulfonylcyclopropanes using
Bakers![]() Rikuhei Tanikaga Noriaki Shibata and Takamitsu Yoneda pg 2253; DOI: 10.1039/a700160f |
Novel ring transformation of nitropyrimidinone; synthetic equivalent of
![]() Nagatoshi Nishiwaki Hui-Ping Wang Kengo Matsuo Yasuo Tohda and Masahiro Ariga pg 2261; DOI: 10.1039/a704354f |
Novel synthesis of substituted
4![]() ![]() ![]() ![]() Reza-Ali Fallahpour and Edwin C. Constable pg 2263; DOI: 10.1039/a704295g |
Catalytic asymmetric epoxidation with a chiral ruthenium porphyrin and
N-oxides
Albrecht Berkessel and Matthias Frauenkron pg 2265; DOI: 10.1039/a704275b |
First diastereoselective [3+2] cycloaddition of chiral
non-racemic alkenyl Fischer carbene complexes with diazomethane
derivatives
José Barluenga Félix Fernández-Marí Argimiro L. Viado Enrique Aguilar and Bernardo Olano pg 2267; DOI: 10.1039/a704228k |
Towards a synthesis of C3-tribenzohemifullerene, a
C42H18 fragment of [60]fullerene
Goverdhan Mehta Gautam Panda Shailesh R. Shah and Ajit C. Kunwar pg 2269; DOI: 10.1039/a702911j |
Butoxycarbonylation of aryl halides catalyzed by a silica-supported
poly[3-(2-cyanoethylsulfanyl)propylsiloxane palladium] complex
Ming-Zhong Cai Cai-Sheng Song and Xian Huang pg 2273; DOI: 10.1039/a702085f |
Remarkable acceleration of a lipase-catalyzed reaction by a thiacrown
ether additive: buffer-free highly regioselective partial hydrolysis of
4-acetoxy-2-methylbut-2-enyl acetate
Toshiyuki Itoh Koichi Mitsukura Kunihiro Kaihatsu Hiroki Hamada Yumiko Takagi and Hiroshi Tsukube pg 2275; DOI: 10.1039/a702894f |
Chromium(II)-mediated synthesis of vinylbis(silanes) from
aldehydes and a study of acid- and base-induced reactions of the derived
epoxybis(silanes): a synthesis of acylsilanes
David M. Hodgson Paul J. Comina and Michael G. B. Drew pg 2279; DOI: 10.1039/a702722b |
Sulfur-controlled 6-exo aryl radical cyclisation of
N-ethenyl-2-(2-bromophenyl)acetamides: synthesis of
()-tetrahydropalmatine and saulatine
Hiroyuki Ishibashi Hirotaka Kawanami Hiroko Nakagawa and Masazumi Ikeda pg 2291; DOI: 10.1039/a702307c |
Synthesis of fused 1,2,5-triazepine-1,5-diones and some N2-
and N3-substituted derivatives: potential conformational
mimetics for cis-peptidyl prolinamides![]() Morag M. Lenman Arwel Lewis and David Gani pg 2297; DOI: 10.1039/a702107k |
Direct C-11 functionalisation of anatoxin-a. Application to the
synthesis of new ligand-based structural probes
Nicholas A. Magnus Laurent Ducry Valérie Rolland Susan Wonnacott and Timothy Gallagher pg 2313; DOI: 10.1039/a702087b |
Oxidative rearrangement and cyclisation of N-substituted
amidines using iodine(III) reagents and the influence of
leaving group on mode of reaction
Christopher A. Ramsden and Helen L. Rose pg 2319; DOI: 10.1039/a702025b |
The synthesis of antioxidants showing selective affinity for low density
lipoproteins
David W. Brown Mary F. Mahon Aleyamma Ninan and Malcolm Sainsbury pg 2329; DOI: 10.1039/a701948c |
Some single electron-transfer reactions of arylimines
David W. Brown Monika Lindquist Mary F. Mahon Bengt Malm Göran N. Nilsson Aleyamma Ninan Malcolm Sainsbury and Christer Westerlund pg 2337; DOI: 10.1039/a701947e |
Zinc(II)-catalysed asymmetric hetero-Diels–Alder
reactions of conjugated dienes with glyoxylate
Sulan Yao Mogens Johannsen and Karl Anker Jørgensen pg 2345; DOI: 10.1039/a701882g |
Lignin–ferulate cross-links in grasses. Part
4.1–3 Incorporation of 5–5-coupled
dehydrodiferulate into synthetic lignin
Stéphane Quideau and John Ralph pg 2351; DOI: 10.1039/a701808h |
Synthesis of glycopeptide sequences of repeating units of the mucins MUC
2 and MUC 3 containing oligosaccharide side-chains with core 1, core 2,
core 3, core 4 and core 6 structure
Nathalie Mathieux Hans Paulsen Morten Meldal and Klaus Bock pg 2359; DOI: 10.1039/a701742a |
Photochemical substitution of halogenopyrrole derivatives
Maurizio D ![]() pg 2369; DOI: 10.1039/a701674c |
Preparation of fluorinated galactosyl nucleoside diphosphates to study
the mechanism of the enzyme galactopyranose
mutase![]() Andrew Burton Paul Wyatt and Geert-Jan Boons pg 2375; DOI: 10.1039/a701630a |
Transglycosylation activity of Bacillus
1,3-1,4-![]() ![]() Josep-Lluís Viladot Vincent Moreau Antoni Planas and Hugues Driguez pg 2383; DOI: 10.1039/a701431g |
Improved, gram scale synthesis of
N,O,O-triacetyl-erythro- and
threo-C18-sphingosines from serine
Alessondro Dondoni Daniela Perrone and Elisa Turturici pg 2389; DOI: 10.1039/a701391d |
Acid-catalyzed rearrangements of flavan-4-phloroglucinol derivatives to
novel
6-hydroxyphenyl-6a,11b-dihydro-6H-[1]benzofuro[2,3-c]
chromenes and hydroxyphenyl-3,2![]() Petrus J. Steynberg Jan P. Steynberg Richard W. Hemingway Daneel Ferreira and G. Wayne McGraw pg 2395; DOI: 10.1039/a700889i |
Synthesis of the marine dibromooxoindoline convolutamydine C
Soyfur Miah Christopher J. Moody Ian C. Richards and Alexandra M. Z. Slawin pg 2405; DOI: 10.1039/a700683g |
Studies towards the synthesis of diazonamide A. Unexpected formation of
a 3,4-bridged indole
Christopher J. Moody Kevin J. Doyle Mark C. Elliott and Timothy J. Mowlem pg 2413; DOI: 10.1039/a700684e |
Reaction of lactim ethers and lactim sulfides with electrophiles: attack
at nitrogen followed by ring-opening under neutral conditions
Mariappan Anbazhagan Arun N. Dixit and Srinivasachari Rajappa pg 2421; DOI: 10.1039/a700523g |
The solid-state diastereoselective formation of oxazolidines
Natalya S. Khruscheva Nikolay M. Loim Viatcheslav I. Sokolov and V. D. Makhaev pg 2425; DOI: 10.1039/a700246g |
Photogeneration of amines from ![]() James F. Cameron C. Grant Willson and Jean M. J. Fréchet pg 2429; DOI: 10.1039/a602018f |
Synthesis of L-selenocystine,
L-[77Se]selenocystine and
L-tellurocystine
Emily M. Stocking Jessie N. Schwarz Hans Senn Michael Salzmann and Louis A. Silks pg 2443; DOI: 10.1039/a600180g |
Nickel-catalysed cross-coupling reactions of aryl halides with
organostannanes
Eiji Shirakawa Kenji Yamasaki and Tamejiro Hiyama pg 2449; DOI: 10.1039/a705078j |
Development of arylhydrazines and diphenyl arylhydrazidophosphates as
photo-induced DNA-cleaving agents
Jih Ru Hwu Chii Shyang Yau Fu Yuan Tsai and Shwu-Chen Tsay pg 2451; DOI: 10.1039/a704706a |
Insertion of ethyl diazoacetate into N–H and S–H bonds
catalyzed by ruthenium porphyrin complexes
Erwan Galardon Paul Le Maux and Gérard Simonneaux pg 2455; DOI: 10.1039/a704687a |
Highly diastereoselective synthesis of densely functionalized
cyclopentanoids by intramolecular azomethine imine cycloadditions
in sugar templates
John K. Gallos Alexandros E. Koumbis and Nicolaos E. Apostolakis pg 2457; DOI: 10.1039/a704207h |
Synthesis of cyclitols fused with a furoxan ring from alditols by
intramolecular nitrile oxide dimerization
John K. Gallos Theoharis V. Koftis Vassiliki I. Karamitrou and Alexandros E. Koumbis pg 2461; DOI: 10.1039/a704208f |
Synthesis of functionalised unsymmetrical diaryliodonium salts
Aneela Shah Victor W. Pike and David A. Widdowson pg 2463; DOI: 10.1039/a704062h |
Glycosylation of silybin
Vladimír K ![]() ![]() ![]() ![]() ![]() pg 2467; DOI: 10.1039/a703283h |
Synthesis of a cis-conformationally restricted peptide bond
isostere and its application to the inhibition of the HIV-1 protease
Andrew D. Abell and Glenn J. Foulds pg 2475; DOI: 10.1039/a702458d |
Synthesis of fused furans by gas-phase pyrolysis of
2-allyloxyarylpropenoic esters![]() Michael Black J. I. G. Cadogan Hamish McNab Andrew D. MacPherson V. Peter Roddam Carol Smith and Helen R. Swenson pg 2483; DOI: 10.1039/a702451g |
Design and preparation of serine–threonine protein phosphatase
inhibitors based upon the nodularin and microcystin toxin structures:
Part 1. Evaluation of key inhibitory features and synthesis of a
rationally stripped-down nodularin macrocycle
Amit P. Mehrotra Kerri L. Webster and David Gani pg 2495; DOI: 10.1039/a702407j |
Design and preparation of serine–threonine protein phosphatase
inhibitors based upon the nodularin and microcystin toxin structures:
Part 2.1 Synthesis of a functionalised nodularin
macrocycle and a stripped-down microcystin macrocycle
Antony B. Maude Amit P. Mehrotra and David Gani pg 2513; DOI: 10.1039/a702410j |
Structures of a new type of yellow pigments, falconensones A and B, from
Emericella falconensis
Nobuko Ogasawara Reiko Mizuno and Ken-ichi Kawai pg 2527; DOI: 10.1039/a701277b |
Asymmetric total synthesis of (+)-carbocyclic uracil polyoxin C
Varinder K. Aggarwal and Nuno Monteiro pg 2531; DOI: 10.1039/a702323e |
Dialkyl phosphonates and tetraalkyl bis(phosphonate)s from the
decomposition of quasi-phosphonium ylidic phosphonates in aqueous
conditions
D. Vaughan Griffiths Khalku Karim and Jayne E. Harris pg 2539; DOI: 10.1039/a702258a |
Reactions of carbene intermediates from the reaction of trialkyl
phosphites with dialkyl benzoylphosphonates: preparation and reactions
of dimethyl
2-(N-tert-butyl-N-methylamino)
benzoylphosphonate and dimethyl 2-(methylamino)benzoylphosphonate
D. Vaughan Griffiths Jayne E. Harris and Belinda J. Whitehead pg 2545; DOI: 10.1039/a701147d |
Stereoselective synthesis of 4-alkoxy-3-methylidenealkanols using
reactions between 2-(1-alkoxyalkyl)propenylstannanes and aldehydes:
X-ray crystal structure of
(1R,4R)-3-methylidene-1-(4-nitrophenyl)pentane-1,4-diol
Pedro Almendros Michelangelo Gruttadauria Madeleine Helliwell and Eric J. Thomas pg 2549; DOI: 10.1039/a702256e |
On the stereoselectivity of reactions of alkoxyallylstannanes and alkoxy
aldehydes
Pedro Almendros and Eric J. Thomas pg 2561; DOI: 10.1039/a702257c |
Synthesis and utilisation of
6-aminotetrahydrobenzo[7]annulenes
David A. Learmonth George R. Proctor and David I. C. Scopes pg 2569; DOI: 10.1039/a702212c |
Palladium-catalysed heteroannulation of vinylic compounds: a highly
convenient method for the synthesis of
N-aryl-1,2,3,4-tetrahydro-1-oxoisoquinoline-3-carboxylic acids
Jyan S. Mahanty Mahuya De and Nitya G. Kundu pg 2577; DOI: 10.1039/a702032e |
Chelation of diamine ligands to zinc porphyrin monolayers amide-linked
to glass
Duncan W. J. McCallien Paul L. Burn and Harry L. Anderson pg 2581; DOI: 10.1039/a701968h |
Synthesis of 2![]() ![]() ![]() Loïc Le Hir de Fallois Jean-Luc Décout and Marc Fontecave pg 2587; DOI: 10.1039/a701820g |
Reaction of trithiazyl trichloride with alkenes and alkynes
Xiao-Guang Duan Xiao-Lan Duan Charles W. Rees and Tai-Yuen Yue pg 2597; DOI: 10.1039/a701818e |
Metal-assisted reactions. Part 27.1
3-Benzyloxy-1,2-benzisothiazole 1,1-dioxide: an unusual ether linkage
that does not permit heterogeneous catalytic hydrogenolysis
Amadeu F. Brigas Pedro M. Goncalves and Robert A. W. Johnstone pg 2603; DOI: 10.1039/a701672g |
Atroposelectivity in the reactions of ortholithiated aromatic tertiary
amides with aldehydes
Peter Bowles Jonathan Clayden Madeleine Helliwell Catherine McCarthy Matthew Tomkinson and Neil Westlund pg 2607; DOI: 10.1039/a701671i |
Synthesis and desaturation of monofluorinated fatty
acids![]() Peter H. Buist Kostas A. Alexopoulos Behnaz Behrouzian Brian Dawson and Bruce Black pg 2617; DOI: 10.1039/a701571b |
Flash vacuum pyrolysis of stabilised phosphorus ylides. Part
10.1 Generation of 2-methylstyrylalkynes and their
thermal cyclisation to 2-alkenylnaphthalenes
R. Alan Aitken Christine Boeters and John J. Morrison pg 2625; DOI: 10.1039/a701427i |
Chiral oximes in asymmetric synthesis. Part 2.1 Addition of
butyllithium to benzaldehyde
O-(1-phenylalkyl)oximes
Peter T. Gallagher James C. A. Hunt Andrew P. Lightfoot and Christopher J. Moody pg 2633; DOI: 10.1039/a700984d |
Synthesis of 1,2-fused indoles by radical cyclisation1 Christopher J. Moody and Claire L. Norton pg 2639; DOI: 10.1039/a700985b |
Asymmetric dihydroxylation of allylic phosphine oxides
Adam Nelson and Stuart Warren pg 2645; DOI: 10.1039/a700374i |
Chemistry of 5-oxodihydroisoxazoles. Part 17.1
Acylation of 5-oxodihydroisoxazoles
Rolf H. Prager Jason A. Smith Ben Weber and Craig M. Williams pg 2659; DOI: 10.1039/a700133i |
Chemistry of 5-oxodihydroisoxazoles. Part 18.1
Synthesis of oxazoles by the photolysis and pyrolysis of
2-acyl-5-oxo-2,5-dihydroisoxazoles
Rolf H. Prager Jason A. Smith Ben Weber and Craig M. Williams pg 2665; DOI: 10.1039/a700134g |
The chemistry of 5-oxodihydroisoxazoles. Part 19.1 The
synthesis and photolysis of
N-thioacylisoxazol-5(2H)-ones
Rolf H. Prager Max R. Taylor and Craig M. Williams pg 2673; DOI: 10.1039/a700646b |
Sodium hydroxide-promoted reaction of 1-substituted
2,3,3-trifluoroprop-1-enyl toluene-p-sulfonates with
alcohols. First efficient and convenient access to
![]() ![]() ![]() Kazumasa Funabiki Chisato Suzuki Seizi Takamoto Masaki Matsui and Katsuyoshi Shibata pg 2679; DOI: 10.1039/a705495e |
Phosphabenzene–rhodium catalysts for the efficient
hydroformylation of terminal and internal olefins
Bernhard Breit Roland Winde and Klaus Harms pg 2681; DOI: 10.1039/a705249i |
Studies in sulfur heterocycles. Part 13.1 An expedient
synthesis of 7-hydroxybenzo[b]thiophene and its 2- and
3-substituted derivatives
Subhendu Sekhar Samanta Sukhen Chandra Ghosh and Asish De pg 2683; DOI: 10.1039/a705119k |
Investigations into nicotinic acetylcholine receptor (nAChR)
antagonists: synthesis of a sub-unit of methyllycaconitine
Lynn C. Baillie John R. Bearder John A. Sherringham and Donald A. Whiting pg 2687; DOI: 10.1039/a704447j |
Phenylselenotris(trimethylsilyl)silane and
phenyltellurotris(trimethylsilyl)silane: versatile reagents for the
preparation of phenylseleno- and phenyltelluro-formates
Carl H. Schiesser and Melissa A. Skidmore pg 2689; DOI: 10.1039/a704402j |
Synthesis of 2,3,4-triphenyl-3-azabicyclo[3.2.0]hepta-1,4-diene and its
novel reaction with dimethyl acetylenedicarboxylate
Kiyoshi Matsumoto Sadahito Goto Naoto Hayashi Takane Uchida and Akikazu Kakehi pg 2691; DOI: 10.1039/a704090c |
One-step syntheses of pyrrolo- and indolo-1,2,5-thiadiazoles and
pyrrolobis[1,2,5]thiadiazoles
Xiao-Guang Duan and Charles W. Rees pg 2695; DOI: 10.1039/a703133e |
[11C]Carbon monoxide in the palladium-mediated synthesis of
11C-labelled ketones
Pelle Lidström Tor Kihlberg and Bengt Långström pg 2701; DOI: 10.1039/a703062b |
Applications of the spiroannulation of tetralins with alkynes; towards
new anti-estrogenic compounds
F. Thomas Boyle Owen Hares Zbigniew S. Matusiak Warren Li and Donald A. Whiting pg 2707; DOI: 10.1039/a702992f |
Carotenoids and related polyenes. Part 4.1 Synthesis of
carotenoid analogues containing a conjugated carbonyl group and their
fluorescence properties
Yumiko Yamano Mamoru Mimuro and Masayoshi Ito pg 2713; DOI: 10.1039/a702815f |
Studies on the reactivity of azetidin-2-ones in phosphate buffer
Nicholas J. Westwood Christopher J. Schofield and Timothy D. W. Claridge pg 2725; DOI: 10.1039/a702673k |
Total synthesis of C31-methyl ketone apocarotenoids. Part
4. First total synthesis of
(3S,5R,6R)-paracentrone
Jarle André Haugan pg 2731; DOI: 10.1039/a702545i |
Antitumour polycyclic acridines. Part 1. Synthesis of
7H-pyrido- and 8H-quino-[4,3,2-kl]acridines
by Graebe–Ullmann thermolysis of 9-(1,2,3-triazol-1-yl)acridines:
application of differential scanning calorimetry to predict optimum
cyclisation conditions
Damien J. Hagan Elena Giménez-Arnau Carl H. Schwalbe and Malcolm F. G. Stevens pg 2739; DOI: 10.1039/a702299i |
Regioselective aryl radical cyclisation. Part 2.1
Synthesis of
octahydro-1H-dibenzo[a,d]cycloheptenes
through 7-endo ring closure
Ajit K. Ghosh Jayanta K. Mukhopadhyaya and Usha Ranjan Ghatak pg 2747; DOI: 10.1039/a702253k |
Enantioselective addition of dialkylzincs to
N-diphenylphosphinylimines using polymer-supported
N,N-dialkylnorephedrines as chiral ligands
Takefumi Suzuki Takanori Shibata and Kenso Soai pg 2757; DOI: 10.1039/a702139i |
Synthesis, structure and reactions of uridine
2![]() ![]() ![]() ![]() Anthony J. Lawrence John B. J. Pavey Mai-Yee Chan Robin A. Fairhurst Stephen P. Collingwood Julie Fisher Richard Cosstick and Ian A. O ![]() pg 2761; DOI: 10.1039/a702088k |
Parasite glycoconjugates. Part 7.1 Synthesis of further
substrate analogues of early intermediates in the biosynthetic pathway
of glycosylphosphatidylinositol membrane anchors
Arthur Crossman Jr John S. Brimacombe and Michael A. J. Ferguson pg 2769; DOI: 10.1039/a701881i |
Stereoselective construction of vicinal diamines. Part
3.1 Routes to the
benz[ f ]indeno[1,7-bc]
azepine and benz[e]indeno[2,1-b][1,4]diazepine ring
systems
Barry S. Orlek and Eleanor A. Crowe pg 2775; DOI: 10.1039/a701762f |
Protection of the guanine residue during synthesis of
2![]() Morten Grøtli Mark Douglas Barbro Beijer Ramon Güimil García Ramon Eritja and Brian Sproat pg 2779; DOI: 10.1039/a700813i |
Design, synthesis and evaluation of a novel series of spiroketals based
on the structure of the antibacterial gyrase inhibitor novobiocin
William Bell Michael H. Block Calum Cook J. Andrew Grant and David Timms pg 2789; DOI: 10.1039/a700647k |
Rapid access to rare natural pyranosides using 1,2-diacetal protected intermediates Steven V. Ley Dafydd R. Owen and Kieron E. Wesson pg 2805; DOI: 10.1039/a705360f |
2-Aminobuta-1,3-dienes as annulation reagents for 4-quinolones and benzothiopyran-4-ones: an attractive route for the highly diastereoselective synthesis of acridine- and thioxanthene-derivatives Uwe Beifuss and Michael Taraschewski pg 2807; DOI: 10.1039/a704289b |
Dimethylsulfonium fluoren-9-ide: solution structure and dynamic behaviour of a semi-stabilised sulfonium ylide Varinder K. Aggarwal Steffen Schade and Brian Taylor pg 2811; DOI: 10.1039/a704010e |
Palladium-catalysed heteroannulation with acetylenic compounds: synthesis of benzofurans1 Nitya G. Kundu Manojit Pal Jyan S. Mahanty and Mahuya De pg 2815; DOI: 10.1039/a703305b |
Ketone homologation to produce ![]() Neil Phillipson Michael S. Anson John G. Montana and Richard J. K. Taylor pg 2821; DOI: 10.1039/a703073h |
Reaction of trithiazyl trichloride with active methylene compounds Xiao-Guang Duan Xiao-Lan Duan and Charles W. Rees pg 2831; DOI: 10.1039/a703033i |
Rapid synthesis of aliphatic amides by reaction of carboxylic acids, Grignard reagent and amines: application to the preparation of [11C]amides Catherine Aubert Cécile Huard-Perrio and Marie-Claire Lasne pg 2837; DOI: 10.1039/a702897k |
Palladium-catalyzed chemoselective intramolecular cyclization of bromoanilinoalkenenitriles Chau-Chen Yang Huo-Mu Tai and Pei-Jiun Sun pg 2843; DOI: 10.1039/a702710i |
Synthesis and conformational analysis of extended calix[4]arenes and a doubly bridged bis-calix[4]arene Mikkel Jørgensen Mogens Larsen Peter Sommer-Larsen Walter Batsberg Petersen and Hanne Eggert pg 2851; DOI: 10.1039/a702610b |
Efficient selective synthesis of 2-substituted indoles from complex-base-promoted arynic cyclisations Catherine Kuehm-Caubère Ivan Rodriguez Bruno Pfeiffer Pierre Renard and Paul Caubère pg 2857; DOI: 10.1039/a702548c |
Aqueous [6+4] cycloadditions of tropone with 1-(glucopyranosyloxy)buta-1,3-diene André Lubineau Giliane Bouchain and Yves Queneau pg 2863; DOI: 10.1039/a702447i |
Unsaturated macrocyclic lactone synthesis via catalytic ring-closing metathesis![]() Konstantinos E. Litinas and Basil E. Salteris pg 2869; DOI: 10.1039/a702353g |
Synthesis of chiral and achiral analogues of ambroxol via palladium-catalysed reactions Anna L. E. Larsson Roberto G. P. Gatti and Jan-E. Bäckvall pg 2873; DOI: 10.1039/a702141k |
Furan-2(3H)- and -2(5H)-ones. Part 8.1 Conformation and di-![]() Osamu Muraoka Genzoh Tanabe Emi Yamamoto Masaru Ono Toshie Minematsu and Takayoshi Kimura pg 2879; DOI: 10.1039/a702108i |
Synthesis and application of ligands for the asymmetric addition of organolithium reagents to imines Catrin A. Jones Iwan G. Jones Mushtaq Mulla Michael North and Lucia Sartori pg 2891; DOI: 10.1039/a702028g |
Fullerene tectonics. Part 1. A programmed precursor to C60 M. John Plater pg 2897; DOI: 10.1039/a701915g |
Fullerene tectonics. Part 2.1 Synthesis and pyrolysis of halogenated benzo[c]phenanthrenes M. John Plater pg 2903; DOI: 10.1039/a701916e |
Use of model cell membranes to demonstrate templated binding of vancomycin group antibiotics Andrew C. Try Gary J. Sharman Robert J. Dancer Ben Bardsley Richard M. H. Entress and Dudley H. Williams pg 2911; DOI: 10.1039/a701880k |
Ring expansions of N-methyl-1,2,5-oxadiazolium and 1,2,3-triazolium perchlorate salts with bases to six-membered azines: direct detection of an addition intermediate in an addition–elimination mechanism and a degradation of 1,2,5-oxadiazolium salts to ![]() Richard N. Butler Elaine C. McKenna John M. McMahon Karen M. Daly Desmond Cunningham and Patrick McArdle pg 2919; DOI: 10.1039/a701233k |
Regioselective synthesis of 6-substituted 2-hydroxybenzaldehyde: efficient synthesis of the immunomodulator tucaresol and related analogues Boulos Zacharie Giorgio Attardo Nancy Barriault and Christopher Penney pg 2925; DOI: 10.1039/a701102d |
Rapid synthesis of polyester dendrimers Zhishan Bo Xi Zhang Changmei Zhang Zhiqiang Wang Meilin Yang Jiacong Shen and Yiping Ji pg 2931; DOI: 10.1039/a700841d |
Simple synthetic entries into the tricyclo[5.3.1.13,9]dodecane and 8-oxatetracyclo[5.4.1.13,10.05,9]tridecane ring systems Weimin Yue Roger Bishop Marcia L. Scudder and Donald C. Craig pg 2937; DOI: 10.1039/a607710b |
Convenient synthesis of cytotoxic (11E)-13-hydroxy-10-oxooctadec-11-enoic acid from undec-10-enoic acid Junzo Nokami Masahiro Osafune Kazuhiro Shiraishi Shin-ichi Sumida and Nobuyuki Imai pg 2947; DOI: 10.1039/a706245a |
Chelation controlled cis-selective acylation of 2-(alkoxycarbonyl)cyclopentylzinc iodides Morio Asaoka Akiko Kosaka Michiko Tanaka Tsuyoshi Ueda Takashi Houkawa and Hisashi Takei pg 2949; DOI: 10.1039/a705554d |
N-Alkylation and [2,3]-sigmatropic rearrangement of N-allyl ![]() Iain Coldham Mark L. Middleton and Philip L. Taylor pg 2951; DOI: 10.1039/a705550a |
Novel stereoselective synthesis of 1,3-dienyl selenides by palladium–copper cocatalyzed cross coupling reactions of (E)-![]() Yun Ma and Xian Huang pg 2953; DOI: 10.1039/a703663i |
A novel, chiral Lewis acid-induced enantioselective hetero Diels–Alder reaction of a thiabutadiene Takao Saito Kayoko Takekawa Jun-ichi Nishimura and Mikako Kawamura pg 2957; DOI: 10.1039/a703590j |
Structural elucidation of trichotetronines: polyketides possessing a bicyclo[2.2.2]octane skeleton with a tetronic acid moiety isolated from Trichoderma sp. Osamu Shirota Vibha Pathak Chowdhury Faiz Hossain Setsuko Sekita Kosuke Takatori and Motoyoshi Satake pg 2961; DOI: 10.1039/a704963c |
Ozone-mediated nitration of adamantane and derivatives with nitrogen dioxide: selectivity in the hydrogen abstraction by nitrogen trioxide and subsequent coupling of the resulting carbon radicals with nitrogen dioxide![]() Hitomi Suzuki and Nobuaki Nonoyama pg 2965; DOI: 10.1039/a704419d |
Synthesis of 5,6-dihydropyrrolo[2,1-a]isoquinolines by rearrangement of 5-methyleneisoxazolidines generated from 1,3-dipolar cycloaddition of 3,4-dihydroisoquinoline N-oxides with allenes: a novel consecutive rearrangement to fused-ring pyrrole derivatives Bao-Xiang Zhao and Shoji Eguchi pg 2973; DOI: 10.1039/a704066k |
Photocyclization of 2-(alkylthio)ethyl benzoylacetates via remote proton transfer following charge-transfer interaction between excited ketone carbonyl and thioether chromophore Yuko Yamazaki Toyoharu Miyagawa and Tadashi Hasegawa pg 2979; DOI: 10.1039/a703825i |
Design, synthesis and antioxidant properties of ovothiol-derived 4-mercaptoimidazoles Vincent Zoete Fabrice Bailly Jean-Pierre Catteau and Jean-Luc Bernier pg 2983; DOI: 10.1039/a703741d |
Displacement of bridgehead sulfonate esters with organometallic reagents: synthesis of 13-alkylated gibberellins Martin Penny Susan M. Westaway and Christine L. Willis pg 2989; DOI: 10.1039/a703587j |
Design, synthesis and pharmacological evaluation of active pyrrole based, nonpeptidic analogues of neurotensin(8-13) Feng Hong Javid Zaidi Yuan-Ping Pang Bernadette Cusack and Elliott Richelson pg 2997; DOI: 10.1039/a703319b |
Azabicyclo[3.2.0]heptan-7-ones (carbapenams) from pyrrole Thomas L. Gilchrist Américo Lemos and Carol J. Ottaway pg 3005; DOI: 10.1039/a703170j |
Rearrangement of cis- and trans-1-methyl-2-(2-thienyl)pyrrolidinium 1-methylides in a non-basic medium Nobuhiko Kawanishi Kazuhiko Fujiwara Naohiro Shirai Yoshiro Sato Keiichiro Hatano and Yukihisa Kurono pg 3013; DOI: 10.1039/a703068a |
C-Glycoside phosphoramidite building block for versatile functionalization of oligodeoxyribonucleotides Jari Hovinen and Harri Salo pg 3017; DOI: 10.1039/a703059b |
v-Triazolines. Part 38.1 New synthesis of 4-aminoquinazolines and 6-aminopurines Emanuela Erba and Daniela Sporchia pg 3021; DOI: 10.1039/a703023a |
Benzoxepine formation by the 1,7 electrocyclisation of diene-conjugated carbonyl ylides: studies on relative rates of cyclisation via intramolecular competition reactions Donal F. O ![]() pg 3025; DOI: 10.1039/a702962d |
Convenient synthesis of 2-alkynyl-cyclopropanes and -oxiranes Mitsuhiro Yoshimatsu Satoshi Gotoh Etsuko Gotoh Genzoh Tanabe and Osamu Muraoka pg 3035; DOI: 10.1039/a702895d |
Influence of a 2-fluoro substituent on diastereoselectivity in the 1,3-dipolar cycloadditions of nitrones Masataka Ihara Yuko Tanaka Nobuyuki Takahashi Yuji Tokunaga and Keiichiro Fukumoto pg 3043; DOI: 10.1039/a702810e |
First synthesis of ortho-trifluoromethylated aryl triflates Feng-Ling Qing Junfa Fan Hong-Bin Sun and Xiang-Jun Yue pg 3053; DOI: 10.1039/a702607b |
Preparation of chiral tricarbonyl arene thiol chromium and its application to asymmetric ring opening of meso-epoxides Shin-ichi Fukuzawa Hirohisa Kato Makoto Ohtaguchi Yuki Hayashi and Hiroshi Yamazaki pg 3059; DOI: 10.1039/a702406a |
Synthesis of functionalised cyclic nitrones via regioselective and unusual [3+2] cycloadditions of ![]() Arun K. Sharma Sujit N. Mazumdar and Mohinder P. Mahajan pg 3065; DOI: 10.1039/a702254i |
Aggregative activation in heterocyclic chemistry. Part 4. Metallation of 2-methoxypyridine: unusual behaviour of the new unimetal superbase BuLi–Me2N(CH2)2OLi (BuLi–LiDMAE) Philippe Gros Yves Fort and Paul Caubère pg 3071; DOI: 10.1039/a701914i |
Regiospecific aromatic chlorination of alkyl phenyl ethers using sodium chlorite catalysed by manganese(III) acetylacetonate and moist alumina in dichloromethane Masao Hirano Shigetaka Yakabe Hiroyuki Monobe James H. Clark and Takashi Morimoto pg 3081; DOI: 10.1039/a701813d |
Solvent-dependent ambident nucleophilicity of phenoxide ion towards nitroporphyrins: synthesis of 2-hydroxyaryl- and 2-aryloxy-5,10,15,20-tetraphenylporphyrins by displacement of a nitro group Maxwell J. Crossley Lionel G. King and Janelle L. Simpson pg 3087; DOI: 10.1039/a701673e |
Model studies towards the synthesis of 4![]() ![]() ![]() ![]() Antonella Leggio Angelo Liguori Loredana Maiuolo Anna Napoli Antonio Procopio Carlo Siciliano and Giovanni Sindona pg 3097; DOI: 10.1039/a701279i |
Remarkable dependence of the regioselectivity of free radical additions to 3-cinnamoyloxazolidin-2-ones on the stability of the intermediate adduct-radical, electrophilicity of the adding radicals and the conditions for their generation Vitali I. Tararov Nikolai Yu. Kuznetzov Vladimir I. Bakhmutov Nikolai S. Ikonnikov Yuri N. Bubnov Victor N. Khrustalev Tatiana F. Saveleva and Yuri N. Belokon pg 3101; DOI: 10.1039/a701154g |
Flash vacuum pyrolysis of stabilised phosphorus ylides. Part 11.1 Unexpected generation and rearrangement of acetyl benzotriazolyl carbene R. Alan Aitken Ian M. Fairhurst Adrian Ford Paul E. Y. Milne Duncan W. Russell and Martin Whittaker pg 3107; DOI: 10.1039/a604594d |
Stereospecific and regioselective catalytic epoxidation of alkenes by a novel ruthenium(II) complex under aerobic conditions Venkitasamy Kesavan and Srinivasan Chandrasekaran pg 3115; DOI: 10.1039/a706729a |
Conjugate Michael-additions with mixed diorganozincs Philip Jones and Paul Knochel pg 3117; DOI: 10.1039/a706637f |
Alkynyl-pyridinium ylid complexes of tungsten(0) and chromium(0): synthesis and cascade insertion reactions Blanca Martín-Vaca and Henri Rudler pg 3119; DOI: 10.1039/a706584a |
A new class of chiral macrocyclic polythiacrown systems and a caveat![]() Mikhail Grabarnik Israel Goldberg and Benzion Fuchs pg 3123; DOI: 10.1039/a706580i |
An efficient total synthesis of ()-laurene Mukund G. Kulkarni and Dhananjay S. Pendharkar pg 3127; DOI: 10.1039/a706510h |
Triphenylphosphine promoted addition of dimethyl acetylenedicarboxylate to 1,2-benzoquinones: facile synthesis of novel ![]() Vijay Nair J. Somarajan Nair A. U. Vinod and Nigam P. Rath pg 3129; DOI: 10.1039/a706272i |
Synthesis of the tetrahydroisoquinoline unit in the AB ring system of the novel antitumor-antibiotic tetrazomine Viviana L. Ponzo and Teodoro S. Kaufman pg 3131; DOI: 10.1039/a706070j |
Selective mono- and bis-condensations of isophthalaldehyde derivative with 6-(o-aminoanilino)cyclodextrins De-Qi Yuan Kahee Fujita Hidefumi Mizushima and Masatoshi Yamaguchi pg 3135; DOI: 10.1039/a705506d |
N-Methyl- and N-benzyl-4-amino[2.2]paracyclophanes as unique planar chiral auxiliaries Andrew Pelter Huw Kidwell and Roger A. N. C. Crump pg 3137; DOI: 10.1039/a705449a |
Novel chemoselective and diastereoselective iron(III)-catalysed Michael reactions of 1,3-dicarbonyl compounds and enones Jens Christoffers pg 3141; DOI: 10.1039/a704873d |
Hexaaza and octaaza macrocycles with 2-hydroxy-3,5-dimethylbenzyl pendant arms S. W. Annie Bligh Nick Choi Evagoras G. Evagorou and Mary McPartlin pg 3151; DOI: 10.1039/a704835a |
Preparation and characterization of 6A-polyamine-mono-substituted ![]() Bruce L. May Suzanna D. Kean Christopher J. Easton and Stephen F. Lincoln pg 3157; DOI: 10.1039/a704467d |
A new synthesis of pyrroles fused with polycyclic skeletons Satoshi Ito Takashi Murashima and Noboru Ono pg 3161; DOI: 10.1039/a704418f |
Studies on pyrazines. Part 34.1 Synthetic approach, stability and tautomerism of 2,6-dihydroxypyrazines Nobuhiro Sato Kaori Matsumoto Masayuki Takishima and Katsura Mochizuki pg 3167; DOI: 10.1039/a704415a |
New precursors for preparing organic conducting materials: synthesis of (R)-hydroxymethylbis(ethylenedithio)tetrathiafulvalene, and the ring expansion of a cyclic sulfate ester Fabien Leurquin Turan Ozturk Melanie Pilkington and John D. Wallis pg 3173; DOI: 10.1039/a704364c |
Stereoselective synthesis of ![]() Hari Babu Mereyala Srinivas Reddy Gurrala and Rajendrakumar Reddy Gadikota pg 3179; DOI: 10.1039/a704310d |
Synthesis, structure and tropicity of an [11][13]fulvalene derivative Gaku Yamamoto Yasuhiro Mazaki Ryoji Kobayashi Hiroyuki Higuchi and J ![]() pg 3183; DOI: 10.1039/a704071g |
Conversion of pyrroles into bi-1,2,5-thiadiazoles: a new route to biheterocycles Xiao-Guang Duan and Charles W. Rees pg 3189; DOI: 10.1039/a704065b |
Regioselective biotransformations of dinitriles using Rhodococcus sp. AJ2701 Otto Meth-Cohn and Mei-Xiang Wang pg 3197; DOI: 10.1039/a703904b |
N-(Diphenylphosphinothioyl)hydroxylamine: preparation, characterisation and base-induced transposition of sulfur and oxygen atoms in its O-benzoyl derivative![]() Martin J. P. Harger pg 3205; DOI: 10.1039/a703695g |
Desilylation of (Z![]() ![]() ![]() ![]() Bianca Flavia Bonini Mauro Comes Franchini Mariafrancesca Fochi Germana Mazzanti and Alfredo Ricci pg 3211; DOI: 10.1039/a703662k |
Efficient synthesis of (6R)-6-amino-1-methyl-4-(3-methylbenzyl)hexahydro-1H-1,4-diazepine from methyl (2R)- and (2S)-1-benzyloxycarbonylaziridine-2-carboxylates Shiro Kato Hiroshi Harada and Toshiya Morie pg 3219; DOI: 10.1039/a703661b |
Preparation of optically active azophenolic crown ethers containing 1-phenylethane-1,2-diol and 2,4-dimethyl-3-oxapentane-1,5-diol as a chiral subunit: temperature-dependent enantiomer selectivity in the complexation with chiral amines![]() Kazuko Ogasahara Keiji Hirose Yoshito Tobe and Koichiro Naemura pg 3227; DOI: 10.1039/a703452k |
Thermodynamically-controlled cyclisation and interconversion of oligocholates: metal ion templated ![]() ![]() Paul A. Brady and Jeremy K. M. Sanders pg 3237; DOI: 10.1039/a703390g |
On the reaction of prop-2-enylidenetriphenylphosphorane derivatives. Novel synthesis of 4,9-methanocyclopentacycloundecene derivatives and their spectroscopic and chemical properties Tohru Takayasu and Makoto Nitta pg 3255; DOI: 10.1039/a703314a |
Azabenzocycloheptenones. Part 20. Synthesis and utilisation of 4-amino-1,2,3,4-tetrahydro-1(1H)-benzazepines Kevin I. Booker-Milburn Ian R. Dunkin Frances C. Kelly Abedawn I. Khalaf David A. Learmonth George R. Proctor and David I. C. Scopes pg 3261; DOI: 10.1039/a703281a |
Synthesis and hybridization properties of ![]() ![]() ![]() ![]() ![]() Pia N. Jørgensen Ulrik S. Sørensen Henrik M. Pfundheller Carl E. Olsen and Jesper Wengel pg 3275; DOI: 10.1039/a703173d |
Synthesis of some novel ![]() Galal H. Elgemeie Ahmed H. Elghandour Ali M. Elzanate and Sayed A. Ahmed pg 3285; DOI: 10.1039/a702343j |
Tetra-n-propylammonium perruthenate (TPAP)-catalysed oxidations of alcohols using molecular oxygen as a co-oxidant Roman Lenz and Steven V. Ley pg 3291; DOI: 10.1039/a707339i |
Enantiospecific total synthesis of (+)-2-pupukeanone Adusumilli Srikrishna and Thumkunta Jagadeeswar Reddy pg 3293; DOI: 10.1039/a706321k |
Stereocontrolled synthesis of ()-![]() Adusumilli Srikrishna and Dange Vijaykumar pg 3295; DOI: 10.1039/a705600a |
Stereoselective epoxidation of electron poor dienes using poly(L-leucine) Joanne V. Allen Michael W. Cappi Pierre D. Kary Stanley M. Roberts Natalie M. Williamson and L. Eduardo Wu pg 3297; DOI: 10.1039/a706238i |
1,5-Asymmetric induction of chirality: highly diastereoselective addition reactions of organoaluminium reagents into ketone groups in the side-chain of ![]() Steven V. Ley Liam R. Cox Graham Meek Karl-Heinz Metten Carmen Piqué and Julia M. Worrall pg 3299; DOI: 10.1039/a704481j |
1,5-Asymmetric induction of chirality: highly diastereoselective synthesis of homoallylic tertiary alcohols by the Lewis acid-mediated addition of allylstannanes into ketones in the side-chain of ![]() Steven V. Ley and Liam R. Cox pg 3315; DOI: 10.1039/a704491g |
1,5-Asymmetric induction of chirality: diastereoselective addition of organoaluminium reagents and allylstannanes into aldehyde groups in the side-chain of ![]() Steven V. Ley Svenja Burckhardt Liam R. Cox and Graham Meek pg 3327; DOI: 10.1039/a704487i |
Regioselective synthesis of bridged azabicyclic compounds using radical translocations/cyclisations of methyl 2-alkynyl-1-(o-iodobenzoyl)pyrrolidine-2-carboxylates: a formal total synthesis of ()-epibatidine Masazumi Ikeda Yasuhiro Kugo Yukari Kondo Taro Yamazaki and Tatsunori Sato pg 3339; DOI: 10.1039/a705226j |
New routes to benzothiophenes, isothiazoles and 1,2,3-dithiazoles Kumaraswamy Emayan Russell F. English Panayiotis A. Koutentis and Charles W. Rees pg 3345; DOI: 10.1039/a704916a |
Enantiospecific syntheses of (R)- and (S)-proline and some derivatives from D-glucono-1,5-lactone Claudio Mazzini Letitia Sambri Henk Regeling Binne Zwanenburg and Gordon J. F. Chittenden pg 3351; DOI: 10.1039/a704915c |
Vinyl glycosides in oligosaccharide synthesis (part 4): glycosidase-catalysed preparation of substituted allyl glycosides Robin R. Gibson Roger P. Dickinson and Geert-Jan Boons pg 3357; DOI: 10.1039/a704703g |
Stereoselective isomerisations of 4-(2![]() ![]() ![]() ![]() Robin G. F. Giles Rodney W. Rickards and Badra S. Senanayake pg 3361; DOI: 10.1039/a704543c |
Synthesis of oligomers related to nylon 6 Gerald M. Brooke Shahid Mohammed and Mark C. Whiting pg 3371; DOI: 10.1039/a704457g |
Synthesis of pyrido[2,3-c]acridines Paul W. Groundwater and Munawar Ali Munawar pg 3381; DOI: 10.1039/a704361i |
Synthesis based on cyclohexadienes. Part 23.1 Total synthesis of 5-epi-pupukean-2-one Krishna Kaliappan and G. S. R. Subba Rao pg 3387; DOI: 10.1039/a704312k |
Synthesis based on cyclohexadienes. Part 24.1 A new total synthesis of pupukean-2-one and a facile entry to copa and ylanga type sesquiterpene skeletons Krishna Kaliappan and G. S. R. Subba Rao pg 3393; DOI: 10.1039/a704314g |
A study on the scope of the photochemical ring contraction of substituted 2-amino-3-cyano-4H-pyrans to cyclobutenes: crystal structure of 3-carbamoyl-3-cyano-1-ethoxycarbonyl-4-isopropyl-2-phenylcyclobutene Diego Armesto Armando Albert Felix H. Cano Nazario Martín Ana Ramos Miriam Rodriguez Jose L. Segura and Carlos Seoane pg 3401; DOI: 10.1039/a703938g |
4,4![]() ![]() ![]() Alistair P. Henderson Jane Riseborough Christine Bleasdale William Clegg Mark R. J. Elsegood and Bernard T. Golding pg 3407; DOI: 10.1039/a703873i |
Enantioselective synthesis of flavonoids. Part 3.1trans- and cis-Flavan-3-ol methyl ether acetates Hendrik van Rensburg Pieter S. van Heerden and Daneel Ferreira pg 3415; DOI: 10.1039/a703316h |
Synthesis of 2![]() ![]() Poul Nielsen Henrik M. Pfundheller Carl Erik Olsen and Jesper Wengel pg 3423; DOI: 10.1039/a703176i |
Epimerization in acid degradation products of artemisinin Shi-Man Hui Koon-Sin Ngo and Geoffrey D. Brown pg 3435; DOI: 10.1039/a702714a |
1,4-Dithiafulvene-substituted ferrocenes and their conversion into extended tetrathiafulvalene electron donors: synthetic, electrochemical and X-ray structural studies Adrian J. Moore Martin R. Bryce Peter J. Skabara Andrei S. Batsanov Leonid M. Goldenberg and Judith A. K. Howard pg 3443; DOI: 10.1039/a702554h |
Switchable electron-rich biindolizine-based macrocycles: synthesis and redox properties T. Kreher H. Sonnenschein B. Costisella and M. Schneider pg 3451; DOI: 10.1039/a702433i |
Studies on bis(2,3![]() David F. Ewing John W. Goodby Sophie Guenais Philippe Letellier Grahame Mackenzie Isabelle Piastrelli and Daniel Plusquellec pg 3459; DOI: 10.1039/a702346d |
Thienothiophenes. Part 2.1 Synthesis, metallation and bromine![]() Lance S. Fuller Brian Iddon and Kevin A. Smith pg 3465; DOI: 10.1039/a701877k |
Steric and electronic effects on the Weiss reaction. Isolation of 1![]() Scott G. Van Ornum Jin Li Greg G. Kubiak and James M. Cook pg 3471; DOI: 10.1039/a701232b |
The X-ray crystal structure, conformation and preparation of anti-3,3,6,6-tetramethylthiepane-4,5-diol: stereochemistry of reduction of a heterocyclic ![]() Neil Feeder Michael J. Ginnelly Ray V. H. Jones Susan OSullivan Stuart Warren and Paul Wyatt pg 3479; DOI: 10.1039/a605572i |
Synthesis of pyridazine fatty ester derivatives in water: a sonochemical approach Marcel S. F. Lie Ken Jie and Prabhavathi Kalluri pg 3485; DOI: 10.1039/a705117d |
Expedient synthesis of lactone analogues of formestane as new potential aromatase inhibitors Elisiário J. Tavares da Silva Maria L. Sá e Melo André S. Campos Neves José A. Paixão L. C. R. Andrade Maria-José M. Almeida and M. M. R. Costa pg 3487; DOI: 10.1039/a705601j |
Oxidation of sulfides to sulfoxides with 3-aryl-2-tert-butyloxaziridines under high pressure Masao Shimizu Isao Shibuya Yoichi Taguchi Satoshi Hamakawa Kunio Suzuki and Takashi Hayakawa pg 3491; DOI: 10.1039/a705022d |
Stereoselective synthesis of (S![]() ![]() ![]() Dawei Ma and Hongqi Tian pg 3493; DOI: 10.1039/a704704e |
Solvent-dependent conformations of a cyclic tetrapeptide Makoto Tamaki Seiji Komiya Mikihiro Yabu Eiji Watanabe Sadatoshi Akabori and Ichiro Muramatsu pg 3497; DOI: 10.1039/a704476c |
Improved procedure for Juli–Colonna asymmetric epoxidation of ![]() ![]() ![]() Brian M. Adger James V. Barkley Sophie Bergeron Michael W. Cappi Benjamin E. Flowerdew Mark P. Jackson Ray McCague Thomas C. Nugent and Stanley M. Roberts pg 3501; DOI: 10.1039/a704413e |
Synthesis of chiral ![]() ![]() Brian L. Booth Nicholas J. Lawrence and Humayan S. Rashid pg 3509; DOI: 10.1039/a703936k |
Stereospecific synthesis of naturally-occurring 4-alkylideneglutamic acids, 4-alkylglutamates and 4-alkylprolines![]() Claire M. Moody and Douglas W. Young pg 3519; DOI: 10.1039/a703489j |
Control of stereochemistry in an intramolecular Diels–Alder reaction by the phenylsulfonyl group; an improved synthesis of pisiferol Edward J. Bush and David W. Jones pg 3531; DOI: 10.1039/a702761c |
On the reaction of azulen-2-ylmethylene(triphenyl)phosphorane. Convenient preparation of azuleno[1,2-f![]() ![]() Tohru Takayasu and Makoto Nitta pg 3537; DOI: 10.1039/a702716h |
An efficient synthesis of novel N-acetyl-3-alkanoyl and 3-dienoyl tetramic acids Margarita Petroliagi and Olga Igglessi-Markopoulou pg 3543; DOI: 10.1039/a702649h |
Structural separation of biological activities of jasmonates and related compounds Siegfried Blechert Christian Bockelmann Oliver Brümmer Martin Füßlein Heidrun Gundlach Georg Haider Swen Hölder Toni M. Kutchan Elmar W. Weiler and Meinhart H. Zenk pg 3549; DOI: 10.1039/a702494k |
Reaction of lithioamino anions with ![]() ![]() Okram Mukherjee Singh Hiriyakkanavar Junjappa and Hiriyakkanavar Ila pg 3561; DOI: 10.1039/a701435j |
Application of PdII-catalysed oxidative cyclisation of hydroxy(vinyl)furan: synthesis of (5R)-diastereomer of (+)-goniofufurone Hari Babu Mereyala Rajendrakumar Reddy Gadikota and Ravikumar Krishnan pg 3567; DOI: 10.1039/a703905k |
A high yield conversion of tetrathiafulvalene into bis(ethylenedithio)tetrathiafulvalene and derivatives Ronald L. Meline and Ronald L. Elsenbaumer pg 3575; DOI: 10.1039/a707814e |
Efficient chemoenzymatic synthesis of (2S,3S![]() ![]() Nitin W. Fadnavis Mohd. Sharfuddin S. Kumara Vadivel and Uday T. Bhalerao pg 3577; DOI: 10.1039/a707507c |
Tandem Wittig–Diels–Alder reaction between sugar-derived phosphoranes and sugar aldehydes. An easy route to optically pure highly oxygenated decalins S ![]() pg 3579; DOI: 10.1039/a707447f |
Pyrolysis of 1-substituted pyrazoles and chloroform at 550C: formation of ![]() Inayat A. Bhatti Reginald E. Busby Murtedza bin Mohamed John Parrick and C. J. Granville Shaw pg 3581; DOI: 10.1039/a705364i |
Competitive reactivity of the aryl isothiocyanate dipolarophile at N![]() ![]() Richard N. Butler Denise C. Grogan Peter D. McDonald and Luke A. Burke pg 3587; DOI: 10.1039/a705233b |
Reactions of the alkyl radical attached to the ring nitrogen of 2-phenylthio-indole, -benzimidazole and -uracil Tomohiro Uetake Mayumi Nishikawa and Masaru Tada pg 3591; DOI: 10.1039/a705139e |
Aggregative activation in heterocyclic chemistry. Part 5.![]() Philippe Gros Yves Fort and Paul Caubère pg 3597; DOI: 10.1039/a705027e |
Preparation of carbocyclic, phosphonate analogues of cyclic adenosine monophosphate (cAMP) Jennifer M. L. Hillman and Stanley M. Roberts pg 3601; DOI: 10.1039/a704961g |
Phosphorus(III) ligands with fluorous ponytails Pravat Bhattacharyya David Gudmunsen Eric G. Hope Ray D. W. Kemmitt Danny R. Paige and Alison M. Stuart pg 3609; DOI: 10.1039/a704872f |
Radical-mediated cyclisation of ![]() ![]() ![]() Joanne F. Jamie and Rodney W. Rickards pg 3613; DOI: 10.1039/a704869f |
Perfluorocarbon fluids as solvent replacements Richard D. Chambers and Andrew R. Edwards pg 3623; DOI: 10.1039/a704823h |
Deracemization of ()-2,3-disubstituted oxiranes via biocatalytic hydrolysis using bacterial epoxide hydrolases: kinetics of an enantioconvergent process Wolfgang Kroutil Martin Mischitz and Kurt Faber pg 3629; DOI: 10.1039/a704812b |
The synthesis of kermesic acid and isokermesic acid derivatives and of related dihydroxyanthraquinones Stephen J. Bingham and John H. P. Tyman pg 3637; DOI: 10.1039/a704317a |
Dirhodium(II)-catalysed intramolecular carbon–hydrogen insertion reaction of ![]() Takayuki Yakura Seiji Yamada Yuka Kunimune Akiharu Ueki and Masazumi Ikeda pg 3643; DOI: 10.1039/a704102k |
Intramolecular photocyclisation reactions of 5-tert-butyldimethylsilyloxymethyl-3-(3-formylpropyl)furan-2(5H![]() David Brown Michael G. B. Drew and John Mann pg 3651; DOI: 10.1039/a703745g |
Syntheses and structures of 3-stannylcholest-5-ene species Heather J. Buchanan Philip J. Cox Solange M. S. V. Doidge-Harrison R. Alan Howie Marcel Jaspars and James L. Wardell pg 3657; DOI: 10.1039/a703596i |
Neurosteroid analogues. Part 5.1 Enantiomers of neuroactive steroids and benz[e]indenes: total synthesis, electrophysiological effects on GABAA receptor function and anesthetic actions in tadpoles Yuefei Hu Lisa L. Wittmer Melissa Kalkbrenner Alex S. Evers Charles F. Zorumski and Douglas F. Covey pg 3665; DOI: 10.1039/a703212i |
Studies in sulfur heterocycles. Part 12.1 Use of 5,6-dihydrobenzo[b]thiophen-7(4H![]() Subhendu Sekhar Samanta Sukhen Chandra Ghosh and Asish De pg 3673; DOI: 10.1039/a702317k |
An unusual carbon–carbon bond scission reaction with molecular oxygen under mild conditions; formation of piperidines from 1-azabicyclo[2.2.2]octanes Timothy Norris Dinos Santafianos and Jon Bordner pg 3679; DOI: 10.1039/a701223c |